SCHEMBL11832003

SCHEMBL11832003

COc1ccc2cc(C(C)O)ccc2n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT2B7 P16662 1/20 0.49
AKR1C3 P42330 3/20 0.40
AKR1C2 P52895 3/20 0.40
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
ABCB11 O95342 1/20 0.38
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CDK6 Q00534 1/20 0.37
PTGS2 P35354 3/20 0.37
PTGS1 P23219 2/20 0.37
TSHR P16473 2/20 0.37
CDC42 P60953 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14288343 0.86 CDK4 (0.41) AKR1C3AKR1C2HDAC3HDAC4HDAC1
SCHEMBL20666274 0.83 CDK4 (0.37) AKR1C3AKR1C2HDAC3HDAC4HDAC1
SCHEMBL11827253 0.81 AKR1C3 (0.61) AKR1C3AKR1C2PTGS2PTGS1TSHR
SCHEMBL23848110 0.81 ABCB11 (0.43) AKR1C3AKR1C2HDAC3HDAC4HDAC1
SCHEMBL11839847 0.80 AKR1C3 (0.37) AKR1C3AKR1C2HDAC3HDAC4HDAC1
SCHEMBL21164372 0.79 BCL2L11 (0.40) AKR1C3AKR1C2HDAC3HDAC4HDAC1
SCHEMBL30134301 0.78 OGA (0.41) UGT2B7CYP11B1CYP11B2CYP1A2LMNA
SCHEMBL30133952 0.78 OGA (0.41) UGT2B7CYP11B1CYP11B2CYP1A2LMNA
SCHEMBL25804159 0.78 OGA (0.41) UGT2B7CYP11B1CYP11B2CYP1A2LMNA
SCHEMBL31201745 0.77 CYP1A2 (0.55) UGT2B7AKR1C3AKR1C2CYP1A2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3991061-A Azanaphthaleneacetic acid derivatives G. D. SEARLE & CO. (US) 1976-11-09 US disclosed