SCHEMBL30133952

SCHEMBL30133952

COc1cnc2ccc(C(C)O)cc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OGA O60502 4/20 0.41
CSF1R P07333 1/20 0.39
NPSR1 Q6W5P4 2/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
UGT2B7 P16662 1/20 0.39
HPGD P15428 4/20 0.38
ALDH1A1 P00352 2/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
NFKB1 P19838 1/20 0.38
HIF1A Q16665 1/20 0.38
GMNN O75496 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
APEX1 P27695 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25804159 1.00 OGA (0.41) OGACSF1RNPSR1NPC1HTT
SCHEMBL30134301 0.94 OGA (0.41) OGACSF1RNPSR1NPC1HTT
SCHEMBL30133769 0.79 OGA (0.43) OGAUGT2B7CYP1A2PLGPLAU
SCHEMBL11832003 0.78 UGT2B7 (0.49) UGT2B7HPGDCYP1A2LMNAMAPT
SCHEMBL30189800 0.77 ALOX5 (0.42) OGACSF1RFGFR2FGFR4FGFR3
SCHEMBL31731081 0.77 CSF1R (0.45) CSF1RNPSR1NPC1HTTRAB9A
SCHEMBL19926730 0.76 CSF1R (0.37) OGACSF1RNPSR1NPC1HTT
SCHEMBL20810404 0.76 CSF1R (0.39) OGACSF1RNPSR1NPC1HTT
SCHEMBL30133963 0.75 OGA (0.40) OGAUGT2B7FGFR2FGFR4FGFR3
SCHEMBL30134314 0.75 UGT2B7 (0.39) OGANPSR1RXFP1UGT2B7HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4658655-A1 CONDENSED HETEROCYCLIC COMPOUNDS AS INHIBITOR OF DIACYLGLYCEROL KINASES Beone Medicines I GmbH (CH) 2025-12-10 EP disclosed
CN-119119033-A Pyrazolopyridone compounds 百济神州有限公司 2024-12-13 CN disclosed
EP-4457224-A1 HETEROCYCLIC COMPOUNDS BeiGene Switzerland GmbH (CH) 2024-11-06 EP disclosed
WO-2024160278-A1 CONDENSED HETEROCYCLIC COMPOUNDS AS INHIBITOR OF DIACYLGLYCEROL KINASES BEIGENE, LTD. (KY) 2024-08-08 WO disclosed
CN-118451073-A Heterocyclic compounds 百济神州有限公司 2024-08-06 CN disclosed
EP-4380936-A1 PYRAZOLOPYRIDINONE COMPOUNDS BeiGene, Ltd. (KY) 2024-06-12 EP disclosed
CN-117836296-A Pyrazolopyridone compounds 百济神州有限公司 2024-04-05 CN disclosed
WO-2023125681-A1 HETEROCYCLIC COMPOUNDS BEIGENE, LTD. (KY) 2023-07-06 WO disclosed
WO-2023011456-A1 PYRAZOLOPYRIDINONE COMPOUNDS BEIGENE, LTD. (KY) 2023-02-09 WO disclosed