SCHEMBL11847697

SCHEMBL11847697

COc1cccc(OC)c1C(C(N)=O)N1CCNCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
ADRB1 P08588 1/20 0.43
DRD2 P14416 1/20 0.43
CYP2C19 P33261 1/20 0.43
DRD3 P35462 1/20 0.43
HTR3A P46098 1/20 0.43
HTR6 P50406 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
SLC6A2 P23975 5/20 0.43
SLC6A4 P31645 5/20 0.43
HTR7 P34969 5/20 0.43
SLC6A3 Q01959 4/20 0.43
KCNH2 Q12809 4/20 0.43
CYP2D6 P10635 3/20 0.43
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
OPRD1 P41143 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4558789 0.86 SLC6A2 (0.48) HTR3EHTR3BADRB1DRD2CYP2C19
SCHEMBL7289950 0.85 SLC6A2 (0.47) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL4559300 0.84 SLC6A4 (0.42) HTR3EHTR3BADRB1DRD2CYP2C19
SCHEMBL2330982 0.81 ADRB1 (0.44) ADRB1HTR3ASLC6A2SLC6A4CYP2D6
SCHEMBL11839058 0.81 ADRB1 (0.44) ADRB1HTR3ASLC6A2SLC6A4CYP2D6
SCHEMBL7289698 0.78 RXFP1 (0.44) HTR3EHTR3BADRB1DRD2CYP2C19
SCHEMBL11850354 0.77 PKM (0.46) OPRD1
SCHEMBL7279547 0.77 PKM (0.46) OPRD1
SCHEMBL7288846 0.76 CHRM2 (0.55) HTR3EHTR3BADRB1CYP2C19HTR3A
SCHEMBL7282505 0.74 TSHR (0.59) ADRB1DRD2CYP2C19DRD3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3987036-A ACYLATION, CORONARY VASODILATORS CASSELLA FARBWERKE MAINKUR AKTIENGESELLSCHAFT (DT) 1976-10-19 US disclosed