SCHEMBL11852811

SCHEMBL11852811

COc1ccc(N(N)CC(C)=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
PARP10 Q53GL7 2/20 0.44
PARP1 P09874 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
PARP4 Q9UKK3 1/20 0.44
MTNR1A P48039 2/20 0.43
MTNR1B P49286 2/20 0.43
MAPT P10636 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ESR2 Q92731 1/20 0.42
NOX1 Q9Y5S8 1/20 0.42
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
HSP90AA1 P07900 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9779992 0.86 KEAP1 (0.56) KEAP1NFE2L2CA1CA2PARP10
SCHEMBL11558445 0.81 MAPT (0.49) KEAP1NFE2L2CA1CA2MTNR1A
SCHEMBL9771242 0.79 ALDH1A1 (0.47) CA2MAPTNPC1TP53RAB9A
SCHEMBL11318899 0.79 KEAP1 (0.41) KEAP1NFE2L2RAB9ASMN1; SMN2CES2
SCHEMBL12656352 0.79 CA1 (0.48) KEAP1NFE2L2CA1CA2PARP10
SCHEMBL15132701 0.78 ALDH1A1 (0.40) MAPTNPC1RAB9AALDH1A1HTT
SCHEMBL8781767 0.77 ALDH1A1 (0.44) MTNR1AMTNR1BNPC1TP53RAB9A
SCHEMBL28904603 0.76 CA1 (0.48) CA1CA2PARP10PARP1PARP2
SCHEMBL2775693 0.75 AOC3 (0.52) CA1CA2MAPTSMN1; SMN2PDK2
SCHEMBL16171362 0.73 SMN1; SMN2 (0.45) KEAP1NFE2L2MTNR1AMTNR1BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3964894-A 1-(FURYL OR THIAZOLYL)CARBONYL-2-METHYL-5-METHOXY-INDOL-3-YL ACETIC ACID CHINOIN GYOGYSZER-ES VEGYESZETI TERMEKEK GYARA RT (HU) 1976-06-22 US disclosed