SCHEMBL11857079

SCHEMBL11857079

O=C(NC1CCNC1)C(c1ccccc1)c1ccccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
CYP1A2 P05177 1/20 0.46
POLB P06746 2/20 0.43
NPY2R P49146 2/20 0.42
KDM1A O60341 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
GAA P10253 1/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
OPRK1 P41145 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CCR1 P32246 1/20 0.39
TLR9 Q9NR96 2/20 0.39
TLR8 Q9NR97 2/20 0.39
TLR7 Q9NYK1 2/20 0.39
C3AR1 Q16581 1/20 0.38
NTRK1 P04629 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159618 0.86 POLB (0.56) ALDH1A1POLBKDM1ACCR1
SCHEMBL23366613 0.84 S1PR1 (0.48) ALDH1A1CYP1A2NPY2RMEN1KMT2A
Hydrochloric Acid SCHEMBL17842193 0.83 S1PR1 (0.47) ALDH1A1CYP1A2NPY2RMEN1KMT2A
SCHEMBL24671897 0.78 POLB (0.53) ALDH1A1POLBKDM1ACCR1
SCHEMBL11226541 0.78 POLB (0.58) ALDH1A1POLBCCR1C3AR1
SCHEMBL11834924 0.77 CCR1 (0.47) ALDH1A1CYP1A2POLBNPY2RGAA
SCHEMBL11839863 0.75 ALDH1A1 (0.45) ALDH1A1CYP1A2POLBNPY2RKDM4E
SCHEMBL11841818 0.74 CYP1A2 (0.50) ALDH1A1CYP1A2POLBNPY2RCCR1
SCHEMBL14477846 0.73 GRM5 (0.63) KMT2AGAAKDM4ENTRK1
SCHEMBL31654175 0.73 GRM5 (0.63) KMT2AGAAKDM4ENTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3984557-A 1-R-3-PYRROLIDINYL-A-PHENYL-A-(2-PYRIDYL) ACETAMIDES, -ACETONITRILES, AND -METHANES A. H. ROBINS COMPANY, INCORPORATED (US) 1976-10-05 US disclosed
US-3984557-A 1-R-3-PYRROLIDINYL-A-PHENYL-A-(2-PYRIDYL) ACETAMIDES, -ACETONITRILES, AND -METHANES A. H. ROBINS COMPANY, INCORPORATED (US) 1976-10-05 US disclosed