SCHEMBL11869205

SCHEMBL11869205

O=C(CCCl)N1Cc2cccc3[nH]cc(c23)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.42
GABRG2 P18507 2/20 0.42
GABRB3 P28472 2/20 0.42
GABRA3 P34903 2/20 0.42
GABRA2 P47869 2/20 0.42
GABRB2 P47870 2/20 0.42
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.40
DRD3 P35462 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
ALDH1A1 P00352 3/20 0.38
KMT2A Q03164 3/20 0.37
GLA P06280 1/20 0.36
MAPK1 P28482 2/20 0.36
NR4A2 P43354 1/20 0.35
PARP1 P09874 1/20 0.35
ROCK1 Q13464 1/20 0.34
KDM4E B2RXH2 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11872266 0.79 NOTUM (0.56) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL24817140 0.77 NOTUM (0.52) DRD2TAAR1ALDH1A1KMT2AMEN1
SCHEMBL29987139 0.77 NOTUM (0.52) DRD2TAAR1ALDH1A1KMT2AMEN1
SCHEMBL4555519 0.72 GABRA1 (0.48) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL11869851 0.72 TMEM97 (0.47) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL11862357 0.71 DRD2 (0.59) DRD2DRD1DRD4DRD5DRD3
Hydrochloric Acid SCHEMBL11858233 0.70 DRD2 (0.58) DRD2DRD1DRD4DRD5DRD3
SCHEMBL741884 0.69 DRD2 (0.48) DRD2DRD1DRD4DRD5DRD3
Hydrochloric Acid SCHEMBL11867318 0.68 DRD2 (0.47) DRD2DRD1DRD4DRD5DRD3
SCHEMBL5385138 0.68 HDAC3 (0.67) TAAR1ALDH1A1KMT2AMAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3950343-A PYRROLOISOQUINOLINE DERIVATIVES AYERST, MCKENNA AND HARRISON LTD. (CA) 1976-04-13 US disclosed