SCHEMBL11889804

SCHEMBL11889804

COC(=O)C=Cc1cccc(NC(=O)c2ccc(N3CCN(C(=O)O)CC3)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
NPC1 O15118 3/20 0.48
RAB9A P51151 2/20 0.48
SNCA P37840 1/20 0.48
MAPT P10636 7/20 0.48
KDM4E B2RXH2 2/20 0.48
TP53 P04637 1/20 0.48
TSHR P16473 1/20 0.48
HSD17B10 Q99714 1/20 0.48
HTT P42858 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HDAC1 Q13547 3/20 0.47
KCNH2 Q12809 2/20 0.47
POLB P06746 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11889803 1.00 PKM (0.51) PKML3MBTL1NPC1RAB9ASNCA
SCHEMBL2452211 0.88 SMN1; SMN2 (0.49) PKML3MBTL1MAPTTP53TSHR
SCHEMBL4134491 0.88 SMN1; SMN2 (0.49) PKML3MBTL1MAPTTP53TSHR
SCHEMBL2452227 0.85 PKM (0.46) PKML3MBTL1NPC1RAB9ASNCA
SCHEMBL2452210 0.85 PKM (0.46) PKML3MBTL1NPC1RAB9ASNCA
SCHEMBL18664648 0.79 PKM (0.60) PKML3MBTL1NPC1RAB9ASNCA
SCHEMBL18664977 0.78 SNCA (0.65) PKML3MBTL1NPC1RAB9ASNCA
SCHEMBL5184275 0.77 MAPT (0.57) PKMNPC1RAB9AMAPTKDM4E
SCHEMBL1535834 0.77 MAPT (0.59) PKML3MBTL1NPC1RAB9AMAPT
Hydrochloric Acid SCHEMBL9409572 0.74 MAPT (0.53) PKML3MBTL1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799663-B1 Modulators of HCV replication ANGELETTI P IST RICHERCHE BIO (IT) 2012-08-01 EP claimed