SCHEMBL11904076

SCHEMBL11904076

C=Cc1cc(C(F)(F)F)nc2c(C(F)(F)F)cccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.46
ADORA2A P29274 5/20 0.46
ADORA1 P30542 5/20 0.46
CYP3A4 P08684 4/20 0.46
ADORA3 P0DMS8 2/20 0.46
CYP2D6 P10635 2/20 0.46
KDM4E B2RXH2 2/20 0.46
ADORA2B P29275 1/20 0.46
CYP2C19 P33261 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
NR1I2 O75469 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
HTR1A P08908 1/20 0.46
TSHR P16473 1/20 0.46
CNR1 P21554 1/20 0.46
GLRA1 P23415 1/20 0.46
SLC6A2 P23975 1/20 0.46
HTR2A P28223 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29441429 1.00 KCNH2 (0.46) KCNH2ADORA2AADORA1CYP3A4ADORA3
SCHEMBL29463858 1.00 KCNH2 (0.46) KCNH2ADORA2AADORA1CYP3A4ADORA3
SCHEMBL1147111 0.85 KCNH2 (0.46) KCNH2ADORA2AADORA1CYP3A4ADORA3
SCHEMBL9541219 0.78 ESR1 (0.41) KCNH2ADORA2AADORA1CYP3A4ADORA3
SCHEMBL1258312 0.78 KCNH2 (0.47) KCNH2ADORA2AADORA1CYP3A4ADORA3
SCHEMBL2790280 0.78 ALDH1A1 (0.48) KCNH2ADORA2AADORA1CYP3A4ADORA3
SCHEMBL2608426 0.76 CYP2D6 (0.46) KCNH2ADORA2AADORA1CYP3A4ADORA3
SCHEMBL1655812 0.76 KCNH2 (0.49) KCNH2ADORA2AADORA1CYP3A4ADORA3
SCHEMBL7689636 0.76 KCNH2 (0.46) KCNH2ADORA2AADORA1CYP3A4ADORA3
SCHEMBL30604781 0.76 KCNH2 (0.46) KCNH2ADORA2AADORA1CYP3A4ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012107532-A1 4-AMINOALCOHOLQUINOLINE DERIVATIVES, ENANTIOSELECTIVE SYNTHESIS METHODS AND THE USE THEREOF Université de Picardie Jules Verne (FR) 2012-08-16 WO claimed
EP-2487157-A1 Enantioselective synthesis method of 4-aminoalcoholquinoline derivatives and the use Université de Picardie Jules Verne (FR) 2012-08-15 EP claimed
WO-2012107532-A1 4-AMINOALCOHOLQUINOLINE DERIVATIVES, ENANTIOSELECTIVE SYNTHESIS METHODS AND THE USE THEREOF Université de Picardie Jules Verne (FR) 2012-08-16 WO disclosed
EP-2487157-A1 Enantioselective synthesis method of 4-aminoalcoholquinoline derivatives and the use Université de Picardie Jules Verne (FR) 2012-08-15 EP disclosed
EP-2487157-A1 Enantioselective synthesis method of 4-aminoalcoholquinoline derivatives and the use Université de Picardie Jules Verne (FR) 2012-08-15 EP disclosed