SCHEMBL11904766

SCHEMBL11904766

Cn1nc(Cc2ccc(Cl)c(Oc3cc(C#N)cc(C(F)F)c3)c2F)n(C)c1=O

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.51
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
KCNH2 Q12809 2/20 0.36
RORC P51449 1/20 0.34
EPAS1 Q99814 3/20 0.33
BRD9 Q9H8M2 1/20 0.31
HTR2A P28223 1/20 0.31
CRHR1 P34998 1/20 0.30
FNTA P49354 1/20 0.30
FNTB P49356 1/20 0.30
PGGT1B P53609 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11904764 0.92 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL11904809 0.92 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL11904782 0.91 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL1653338 0.91 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL11904806 0.90 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL11904686 0.89 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19KCNH2EPAS1
SCHEMBL11904765 0.89 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19KCNH2EPAS1
SCHEMBL5178143 0.88 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL4810352 0.87 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL1652202 0.85 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19KCNH2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773790-B1 BENZYLTRIAZOLONE COMPOUNDS AS NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2012-08-15 EP claimed