SCHEMBL11904809

SCHEMBL11904809

Cn1nc(Cc2ccc(Cl)c(Oc3cc(C#N)cc(C#N)c3)c2F)n(C)c1=O

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.56
CYP2C9 P11712 2/20 0.55
CYP2C19 P33261 2/20 0.55
KCNH2 Q12809 5/20 0.39
BRD9 Q9H8M2 1/20 0.35
HTR2A P28223 2/20 0.34
EPAS1 Q99814 4/20 0.33
RORC P51449 1/20 0.32
NPBWR1 P48145 1/20 0.32
MCHR1 Q99705 1/20 0.32
SLC6A4 P31645 1/20 0.32
CRHR1 P34998 1/20 0.32
BRAF P15056 1/20 0.31
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11904765 0.95 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19KCNH2BRD9
SCHEMBL11904766 0.92 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19KCNH2BRD9
SCHEMBL11904807 0.91 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL11904215 0.89 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL11904762 0.87 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19KCNH2BRD9
SCHEMBL5180307 0.86 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL11903899 0.85 CYP3A4 (0.59) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL4800446 0.85 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19KCNH2HTR2A
SCHEMBL11904764 0.84 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19KCNH2EPAS1
SCHEMBL2347420 0.83 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19KCNH2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773790-B1 BENZYLTRIAZOLONE COMPOUNDS AS NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2012-08-15 EP claimed