SCHEMBL11971072

SCHEMBL11971072

Cc1nc(-c2cnn(C)c2Br)c2c(=O)[nH]cnn12

nearest known ligand 0.48

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 17/20 0.48
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11971200 0.80 PDE2A (0.59) PDE2A
SCHEMBL11971146 0.76 PDE2A (0.64) PDE2A
SCHEMBL11971301 0.75 ALDH1A1 (0.38) PDE2AALDH1A1
SCHEMBL16210100 0.75 BRD4 (0.46) PDE2A
SCHEMBL16210384 0.74 PDE2A (0.38) PDE2AALDH1A1
SCHEMBL11971379 0.74 PDE2A (0.44) PDE2A
SCHEMBL16210056 0.73 PDE10A (0.44) PDE2A
SCHEMBL11971560 0.73 PDE2A (0.49) PDE2A
SCHEMBL11971375 0.73 PDE2A (0.65) PDE2A
SCHEMBL18742167 0.71 PDE2A (0.40) PDE2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9200000-B2 Imidazo[5,1-f][1,2,4]triazines for the treatment of neurological disorders PFIZER INC. (US) 2015-12-01 US disclosed
US-9200000-B2 Imidazo[5,1-f][1,2,4]triazines for the treatment of neurological disorders PFIZER INC. (US) 2015-12-01 US disclosed
US-9200000-B2 Imidazo[5,1-f][1,2,4]triazines for the treatment of neurological disorders PFIZER INC. (US) 2015-12-01 US disclosed
US-20140066622-A1 Imidazo[5,1-f][1,2,4]Triazines For The Treatment of Neurological Disorders PFIZER INC. (US) 2014-03-06 US disclosed
US-20140066622-A1 Imidazo[5,1-f][1,2,4]Triazines For The Treatment of Neurological Disorders PFIZER INC. (US) 2014-03-06 US disclosed
US-20140066622-A1 Imidazo[5,1-f][1,2,4]Triazines For The Treatment of Neurological Disorders PFIZER INC. (US) 2014-03-06 US disclosed
US-8598155-B2 Imidazo[5,1-f][1,2,4]triazines for the treatment of neurological disorders PFIZER INC. (US) 2013-12-03 US disclosed
US-20120214791-A1 Imidazo[5,1-f][1,2,4]Triazines for the Treatment of Neurological Disorders PFIZER INC. 2012-08-23 US disclosed
US-20120214791-A1 Imidazo[5,1-f][1,2,4]Triazines for the Treatment of Neurological Disorders PFIZER INC. 2012-08-23 US disclosed
US-20120214791-A1 Imidazo[5,1-f][1,2,4]Triazines for the Treatment of Neurological Disorders PFIZER INC. 2012-08-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140066622-A1 Imidazo[5,1-f][1,2,4]Triazines For The Treatment of Neurological Disorders GRIK5, GRIN2C, BDNF PDE2A 1800/4885ALDH1A1 545/4885
US-20120214791-A1 Imidazo[5,1-f][1,2,4]Triazines for the Treatment of Neurological Disorders GRIK5, GRIN2C, BDNF PDE2A 1800/4885ALDH1A1 545/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.