SCHEMBL11983073

SCHEMBL11983073

Cc1nc2cccc(Br)c2cc1Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MEN1 O00255 3/20 0.42
CYP1A2 P05177 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
TP53 P04637 1/20 0.41
GPR3 P46089 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 2/20 0.40
BACE1 P56817 1/20 0.40
KDM4E B2RXH2 1/20 0.40
STAT3 P40763 1/20 0.40
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
GAA P10253 1/20 0.38
TLR8 Q9NR97 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29923867 0.84 GRM1 (0.45) SMN1; SMN2CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL24915844 0.84 GRM1 (0.45) SMN1; SMN2CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL11982911 0.81 KMT2A (0.42) KMT2ASMN1; SMN2MEN1CYP1A2NPSR1
SCHEMBL13227179 0.81 MAPK1 (0.43) CYP1A2CYP3A4CYP2C9L3MBTL1
SCHEMBL13227169 0.80 SMN1; SMN2 (0.55) KMT2ASMN1; SMN2MEN1CYP1A2NPSR1
SCHEMBL24916325 0.80 BACE1 (0.47) KMT2ACYP1A2GPR3ALDH1A1HPGD
SCHEMBL29923623 0.80 BACE1 (0.47) KMT2ACYP1A2GPR3ALDH1A1HPGD
SCHEMBL11982989 0.77 GRM1 (0.39) SMN1; SMN2CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7253268 0.71 CYP1A2 (0.63) KMT2ASMN1; SMN2MEN1CYP1A2CYP2C19
SCHEMBL24915779 0.71 MAPT (0.45) KMT2ASMN1; SMN2MEN1NPSR1GPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1898914-B1 QUINOLINE DERIVATIVES AS ANTIBACTERIAL AGENTS JANSSEN PHARMACEUTICA NV (BE) 2012-08-15 EP disclosed