SCHEMBL29923867

SCHEMBL29923867

CCc1cc2c(Br)cccc2nc1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 2/20 0.45
BACE1 P56817 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
GPR3 P46089 1/20 0.39
GABRA1 P14867 1/20 0.38
GABRB2 P47870 1/20 0.38
MAPK1 P28482 1/20 0.38
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ELANE P08246 1/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
NUDT1 P36639 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24915844 1.00 GRM1 (0.45) GRM1BACE1CYP1A2CYP2D6CYP2C9
SCHEMBL11983073 0.84 KMT2A (0.42) BACE1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL29923623 0.79 BACE1 (0.47) BACE1CYP1A2GPR3MAPTALDH1A1
SCHEMBL24916325 0.79 BACE1 (0.47) BACE1CYP1A2GPR3MAPTALDH1A1
SCHEMBL24915592 0.78 GRM1 (0.43) GRM1CYP1A2CYP2C9GPR3MAPK1
SCHEMBL24916496 0.77 BACE1 (0.42) BACE1CYP1A2MAPK1MAPTNPC1
SCHEMBL29923622 0.77 BACE1 (0.42) BACE1CYP1A2MAPK1MAPTNPC1
SCHEMBL29923988 0.73 MAPT (0.45) BACE1RXFP1GPR3MAPTNPC1
SCHEMBL24915779 0.73 MAPT (0.45) BACE1RXFP1GPR3MAPTNPC1
SCHEMBL13029622 0.73 ALDH1A1 (0.55) GRM1CYP1A2MAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed