Naringin

Naringin

SCHEMBL1201445

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nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 1.00
GSK3B P49841 2/20 1.00
CYP19A1 P11511 2/20 1.00
UBE2N P61088 1/20 1.00
PKM P14618 1/20 0.88
SLCO2B1 O94956 2/20 0.79
XDH P47989 2/20 0.73
SYNJ2 O15056 1/20 0.69
KDM1A O60341 2/20 0.66
DPP4 P27487 1/20 0.66
TDP1 Q9NUW8 2/20 0.62
POLB P06746 1/20 0.62
CALM1 P0DP23 1/20 0.62
CACNA1B Q00975 1/20 0.62
APBA1 Q02410 1/20 0.62
CTDSP1 Q9GZU7 1/20 0.62
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
TRPA1 O75762 1/20 0.57
P4HB P07237 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Naringin SCHEMBL30073709 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM
Naringin SCHEMBL20383126 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM
Naringin SCHEMBL16656151 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM
Naringin SCHEMBL20386954 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM
Naringin SCHEMBL2614060 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM
Naringin SCHEMBL16592383 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM
Naringin SCHEMBL13237107 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM
Naringin SCHEMBL23431 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM
Naringin SCHEMBL14114613 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM
Naringin SCHEMBL30383784 1.00 PTPN1 (1.00) PTPN1GSK3BCYP19A1UBE2NPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120924-B1 AN ANTI-DIABETIC EXTRACT OF HONEYBUSH ZADEC APS (DK) 2016-03-09 EP disclosed
CN-104706855-A Preparation methods and application of Jichuan decoction traditional Chinese medicine extract JIANGSU HAIWANG HEALTH BIOLOG SCIENCE & TECHNOLOGY CO LTD 2015-06-17 CN disclosed
US-20120251643-A1 ANTI-DIABETIC EXTRACT OF HONEYBUSH ZADEC APS (DK) 2012-10-04 US disclosed
US-20110045108-A1 ANTI-DIABETIC EXTRACT OF HONEYBUSH ZADEC APS (DK) 2011-02-24 US disclosed
EP-2120924-A2 AN ANTI-DIABETIC EXTRACT OF HONEYBUSH Zadec APS (DK) 2009-11-25 EP disclosed
WO-2008110552-A9 AN ANTI-DIABETIC EXTRACT OF HONEYBUSH ZADEC APS (DK) 2008-12-04 WO disclosed
WO-2008110552-A2 AN ANTI-DIABETIC EXTRACT OF HONEYBUSH ZADEC APS (DK) 2008-09-18 WO disclosed
US-20040038914-A1 Flavone/ flavanone derivatives for the systemic treatment and prophlaxis of uv-induced dermatoses KRUTMANN JEAN (DE) 2004-02-26 US disclosed
EP-1085865-A1 USE OF CYTOPROTECTANTS Seglen, Per (NO) 2001-03-28 EP disclosed
WO-2000000191-A1 USE OF CYTOPROTECTANTS SEGLEN PER (NO) 2000-01-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110045108-A1 ANTI-DIABETIC EXTRACT OF HONEYBUSH IAPP, DPP4, DPP3 PTPN1 2676/4885GSK3B 1949/4885CYP19A1 4557/4885
US-20120251643-A1 ANTI-DIABETIC EXTRACT OF HONEYBUSH IAPP, DPP4, DPP3 PTPN1 2676/4885GSK3B 1949/4885CYP19A1 4557/4885
US-20040038914-A1 Flavone/ flavanone derivatives for the systemic treatment and prophlaxis of uv-induced dermatoses COLGALT1, PNN, F2 PTPN1 2605/4885GSK3B 2515/4885CYP19A1 85/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.