SCHEMBL12018902

SCHEMBL12018902

CCc1cc(O)c(C(=O)OC)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
HSD17B10 Q99714 4/20 0.44
TSHR P16473 3/20 0.44
KDM4E B2RXH2 3/20 0.44
HPGD P15428 2/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
GSK3B P49841 1/20 0.42
GAA P10253 3/20 0.41
MAPK1 P28482 2/20 0.41
MAPT P10636 5/20 0.41
KMT2A Q03164 5/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
POLB P06746 2/20 0.40
XDH P47989 2/20 0.40
LMNA P02545 1/20 0.40
NFKB1 P19838 1/20 0.40
GFER P55789 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9826082 0.86 HSD17B10 (0.49) ALDH1A1HSD17B10TSHRKDM4EHPGD
SCHEMBL10266096 0.81 ALDH1A1 (0.46) ALDH1A1HSD17B10TSHRKDM4EHPGD
SCHEMBL10068646 0.81 ALDH1A1 (0.47) ALDH1A1HSD17B10TSHRKDM4EHPGD
SCHEMBL9529269 0.76 TSHR (0.45) ALDH1A1HSD17B10TSHRKDM4EHPGD
SCHEMBL7670938 0.76 TSHR (0.45) ALDH1A1HSD17B10TSHRKDM4EHPGD
SCHEMBL577650 0.76 MAPT (0.45) ALDH1A1HSD17B10TSHRKDM4EHPGD
SCHEMBL17203079 0.75 GSK3B (0.52) ALDH1A1KDM4EHPGDGSK3BGAA
SCHEMBL11522285 0.74 MAPT (0.49) HSD17B10TSHRKDM4EHPGDGSK3B
SCHEMBL577651 0.74 MAPT (0.44) ALDH1A1HSD17B10TSHRKDM4EHPGD
SCHEMBL1374020 0.74 TSHR (0.44) HSD17B10TSHRKDM4EHPGDGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019826-B1 THIOPHENE-CARBOXAMIDES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2012-08-29 EP disclosed