Perospirone

Perospirone

SCHEMBL120579

O=C1[C@H]2CCCC[C@H]2C(=O)N1CCCCN1CCN(c2nsc3ccccc23)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 1.00
LMNA P02545 1/20 1.00
CHRM2 P08172 1/20 1.00
ADRA2A P08913 1/20 1.00
CHRM1 P11229 1/20 1.00
DRD1 P21728 1/20 1.00
TBXA2R P21731 1/20 1.00
SLC6A2 P23975 1/20 1.00
SLC6A4 P31645 1/20 1.00
ADRA1A P35348 1/20 1.00
OPRM1 P35372 1/20 1.00
DRD3 P35462 1/20 1.00
SLC6A3 Q01959 1/20 1.00
KCNH2 Q12809 1/20 1.00
DRD2 P14416 5/20 0.73
HTR2A P28223 5/20 0.73
HTR7 P34969 4/20 0.73
HTR6 P50406 4/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Perospirone SCHEMBL6691734 1.00 HTR1A (1.00) HTR1ALMNACHRM2ADRA2ACHRM1
Perospirone SCHEMBL30061058 1.00 HTR1A (1.00) HTR1ALMNACHRM2ADRA2ACHRM1
Perospirone SCHEMBL29846330 0.99 HTR1A (0.98) HTR1ALMNACHRM2ADRA2ACHRM1
Perospirone SCHEMBL1155757 0.99 HTR1A (0.98) HTR1ALMNACHRM2ADRA2ACHRM1
Perospirone SCHEMBL28506465 0.99 HTR1A (0.98) HTR1ALMNACHRM2ADRA2ACHRM1
Perospirone SCHEMBL1651000 0.98 HTR1A (0.96) HTR1ALMNACHRM2ADRA2ACHRM1
Perospirone SCHEMBL1865565 0.98 HTR1A (0.96) HTR1ALMNACHRM2ADRA2ACHRM1
Perospirone SCHEMBL5435087 0.98 HTR1A (0.96) HTR1ALMNACHRM2ADRA2ACHRM1
Perospirone SCHEMBL28054292 0.94 HTR1A (0.89) HTR1ALMNACHRM2ADRA2ACHRM1
SCHEMBL7283429 0.88 HTR1A (0.79) HTR1ALMNACHRM2ADRA2ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3358 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12527754-B2 Methods and compositions for preventing and treating metabolic syndrome induced by antipsychotic treatment and related diseases and conditions TUFTS MEDICAL CENTER, INC. (US) 2026-01-20 US claimed
EP-4674482-A2 PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF Otsuka Pharmaceutical Co., Ltd. (JP) 2026-01-07 EP claimed
US-20250367212-A1 PHARMACOTHERAPY FOR OBSESSIVE-COMPULSIVE DISORDER TARGETING DOPAMINE D1 SIGNAL IN STRIATAL STRIOSOMES MATSUMOTO SHINICHI (JP) 2025-12-04 US claimed
US-20250333792-A1 GENE PANEL FOR IDENTIFYING HYPO SEPSIS PHENOTYPE PATIENTS UNIV FLORIDA (US) 2025-10-30 US claimed
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS INC (US) 2025-09-25 US claimed
EP-4618973-A1 METHODS OF SWITCHING NEUROPSYCHIATRIC MEDICATIONS USING ULOTARONT Sumitomo Pharma America, Inc. (US) 2025-09-24 EP claimed
US-20250235443-A1 USE OF ROLUPERIDONE TO TREAT NEGATIVE SYMPTOMS AND DISORDERS, INCREASE NEUROPLASTICITY, AND PROMOTE NEUROPROTECTION MINERVA NEUROSCIENCES, INC. 2025-07-24 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
EP-4558622-A1 METHODS AND COMPOSITIONS FOR GENERATING HUMAN MIDBRAIN DOPAMINERGIC NEURONS FROM NEURAL PROGENITOR CELLS Trailhead Biosystems Inc. (US) 2025-05-28 EP claimed
WO-2025101418-A1 TREATMENT OF PSYCHIATRIC OR NEUROLOGICAL DISORDERS IN PATIENTS WITH PROMINENT ANHEDONIA USING IRDABISANT AS A MONOTHERAPY OR IN COMBINATION WITH AN ANTIPSYCHOTIC AGENT ALTO NEUROSCIENCE, INC. (US) 2025-05-15 WO claimed
EP-1238676-B1 Combination of a serotonin reuptake inhibitor and an atypical antipsychotic for use in depression, obsessive compulsive disorder and psychosis PFIZER PROD INC (US) 2004-05-19 EP claimed
EP-1404342-A1 TREATMENT OF PSYCHOTIC DISORDERS COMPRISING CO-THERAPY WITH ANTICONVULSANT DERIVATIVES AND ATYPICAL ANTIPSYCHOTICS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-04-07 EP claimed
EP-1353675-A2 NEW DRUG COMBINATIONS OF NOREPINEHRINE REUPTAKE INHIBITORS AND NEUROLEPTIC AGENTS PHARMACIA & UPJOHN COMPANY (US) 2003-10-22 EP claimed
WO-2003066039-A1 COMBINATION THERAPY FOR TREATMENT OF SCHIZOPHRENIA ABBOTT LABORATORIES (US) 2003-08-14 WO claimed
US-20030109546-A1 Treatment of psychotic disorders comprising co-therapy with anticonvulsant derivatives and atypical antipsychotics ORTHO-MCNEIL PHARMACEUTICAL, INC. 2003-06-12 US claimed
WO-2002087590-A1 TREATMENT OF PSYCHOTIC DISORDERS COMPRISING CO-THERAPY WITH ANTICONVULSANT DERIVATIVES AND ATYPICAL ANTIPSYCHOTICS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2002-11-07 WO claimed
US-20020156067-A1 New drug combinations PHARMACIA & UPJOHN COMPANY 2002-10-24 US claimed
EP-1238676-A1 Combination of a serotonin reuptake inhibitor and an atypical antipsychotic for use in depression, obsessive compulsive disorder and psychosis Pfizer Products Inc. (US) 2002-09-11 EP claimed
US-20020123490-A1 Combination treatment for anxiety, depression, obsessive compulsive disorder and psychosis PFIZER INC. 2002-09-05 US claimed
WO-2002053140-A2 NEW DRUG COMBINATIONS OF NOREPINEHRINE REUPTAKE INHIBITORS AND NEUROLEPTIC AGENTS PHARMACIA & UPJOHN COMPANY (US) 2002-07-11 WO claimed