SCHEMBL12067985

SCHEMBL12067985

CC(C)(C)CCNS(=O)(=O)c1ccc(C(=O)O)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
TDP1 Q9NUW8 3/20 0.40
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
HTT P42858 2/20 0.39
CA12 O43570 3/20 0.38
CA9 Q16790 3/20 0.38
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ESR1 P03372 1/20 0.36
POLB P06746 1/20 0.36
NR4A1 P22736 1/20 0.36
APEX1 P27695 1/20 0.36
RECQL P46063 1/20 0.36
DUSP3 P51452 1/20 0.36
PTPN5 P54829 1/20 0.36
PTPN11 Q06124 1/20 0.36
ESR2 Q92731 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12067161 0.84 CA12 (0.50) ALDH1A1TDP1HTTCA12CA9
SCHEMBL12066716 0.80 ALDH1A1 (0.42) ALDH1A1TDP1HTTCYP2C9CYP2C19
SCHEMBL26144895 0.77 TDP1 (0.45) ALDH1A1TDP1HTTCYP2C9CYP2C19
SCHEMBL15625510 0.72 TDP1 (0.46) ALDH1A1TDP1HTTCYP2C9CYP2C19
SCHEMBL3410883 0.70 HTT (0.54) ALDH1A1TDP1HTTCYP2C9CYP2C19
SCHEMBL24462107 0.70 TDP1 (0.50) ALDH1A1TDP1HTTESR1POLB
SCHEMBL8473107 0.70 HTT (0.48) ALDH1A1HTTCA12CA9CYP2C9
SCHEMBL568367 0.69 TDP1 (0.53) ALDH1A1TDP1HTTESR1POLB
SCHEMBL17286586 0.69 ALDH1A1 (0.46) ALDH1A1TDP1HTTCYP2C9CYP2C19
SCHEMBL2007731 0.69 HTT (0.63) ALDH1A1TDP1HTTCA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149841-A1 SUBSTITUTED THIAZOLIDINEDIONE INDAZOLES, INDOLES AND BENZOTRIAZOLES AS ESTROGEN-RELATED RECEPTOR-α MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-12-01 WO disclosed