SCHEMBL12090791

SCHEMBL12090791

CCc1cc(F)c(CC)nc1Cl

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
PSMB5 P28074 1/20 0.31
GLA P06280 1/20 0.31
HTT P42858 1/20 0.31
CRHR1 P34998 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
CTRC Q99895 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
GRM1 Q13255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8235127 0.83 KEAP1 (0.47) KEAP1NFE2L2SMN1; SMN2ESR1ESR2
SCHEMBL4131119 0.79
SCHEMBL13082503 0.78 DHFR (0.33) GLAHTTSMN1; SMN2CYP1A2CYP3A4
SCHEMBL4180064 0.77 KEAP1 (0.64) KEAP1NFE2L2SMN1; SMN2
SCHEMBL6050406 0.74 KHK (0.57) GLAHTTSMN1; SMN2CYP1A2CYP2C9
SCHEMBL12090790 0.74 SMN1; SMN2 (0.31) SMN1; SMN2
SCHEMBL30047831 0.71 KEAP1 (0.39) KEAP1NFE2L2GLAHTTSMN1; SMN2
SCHEMBL13082588 0.71 KEAP1 (0.35) KEAP1NFE2L2GLAHTTSMN1; SMN2
SCHEMBL14047371 0.69 DRD4 (0.43) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL27883300 0.69 KDM4E (0.33) HTTSMN1; SMN2ESR1ESR2GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367831-B2 Heterocyclic compound or salt thereof and intermediate thereof TOYAMA CHEMICAL CO., LTD. (JP) 2013-02-05 US disclosed
US-20120226035-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-09-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120226035-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF IKZF3, ZC3HAV1L, CXXC5 KEAP1 853/4885NFE2L2 1532/4885PSMB5 1143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.