Dexfenfluramine

Dexfenfluramine

SCHEMBL120916

CCN[C@@H](C)Cc1cccc(C(F)(F)F)c1.Cl

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7

The experimentally established mechanism targets of Dexfenfluramine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A known ✓ P28223 4/20 0.97
HTR2B known ✓ P41595 4/20 0.97
HTR2C known ✓ P28335 4/20 0.62
HTR1A known ✓ P08908 2/20 0.56
HTR1D known ✓ P28221 1/20 0.45
HTR7 known ✓ P34969 1/20 0.45
HTR5A known ✓ P47898 1/20 0.45
HTR6 known ✓ P50406 1/20 0.45
SLC6A4 P31645 6/20 0.97
SIGMAR1 Q99720 4/20 0.97
ADRA2C P18825 4/20 0.97
DRD3 P35462 4/20 0.97
ADRA1A P35348 2/20 0.97
OPRK1 P41145 2/20 0.97
LMNA P02545 1/20 0.97
MAPT P10636 1/20 0.97
CYP3A4 P08684 3/20 0.65
CYP2D6 P10635 3/20 0.65
CYP1A2 P05177 2/20 0.65
TP53 P04637 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fenfluramine SCHEMBL11140094 1.00 SLC6A4 (0.97) SLC6A4SIGMAR1HTR2AHTR2BADRA2C
Levofenfluramine SCHEMBL30951308 1.00 SLC6A4 (0.97) SLC6A4SIGMAR1HTR2AHTR2BADRA2C
Dexfenfluramine SCHEMBL29362838 1.00 SLC6A4 (0.97) SLC6A4SIGMAR1HTR2AHTR2BADRA2C
Fenfluramine SCHEMBL6276588 1.00 SLC6A4 (0.97) SLC6A4SIGMAR1HTR2AHTR2BADRA2C
Fenfluramine SCHEMBL39491 1.00 SLC6A4 (0.97) SLC6A4SIGMAR1HTR2AHTR2BADRA2C
Fenfluramine SCHEMBL9080932 1.00 SLC6A4 (0.97) SLC6A4SIGMAR1HTR2AHTR2BADRA2C
Fenfluramine SCHEMBL9276141 1.00 SLC6A4 (0.97) SLC6A4SIGMAR1HTR2AHTR2BADRA2C
Fenfluramine SCHEMBL10947502 0.98 SLC6A4 (0.94) SLC6A4SIGMAR1HTR2AHTR2BADRA2C
Fenfluramine SCHEMBL10602733 0.98 SLC6A4 (0.94) SLC6A4SIGMAR1HTR2AHTR2BADRA2C
Fenfluramine SCHEMBL20590765 0.98 SLC6A4 (0.94) SLC6A4SIGMAR1HTR2AHTR2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6342 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120138634-A Environment-friendly efficient polishing and freckle-developing process for brass artware 广州番禺职业技术学院 2025-06-13 CN claimed
CN-118924651-B Composition with anti-dandruff effect and preparation method thereof 珑玥实业(广州)有限公司 2025-01-24 CN claimed
CN-119059878-A High-carbon isomeric alcohol for preparing aviation fuel and preparation method thereof 广东工业大学 2024-12-03 CN claimed
CN-119028481-A Method for constructing vector prediction model of dissolved organic matter isomeride based on graph learning 香港科技大学深圳研究院 2024-11-26 CN claimed
CN-118930404-A Method for optimizing butanol and octanol product structure 天津渤化永利化工股份有限公司 2024-11-12 CN claimed
CN-118831531-A Method and system for producing paraxylene by using low-carbon aromatic hydrocarbon 中国石化工程建设有限公司 2024-10-25 CN claimed
CN-118813219-A Temperature-resistant salt-resistant anti-swelling clay stabilizer and preparation process and application thereof 北京弘毅恩泽能源技术有限公司 2024-10-22 CN claimed
CN-115772067-B Purification method of high-reflection-type special hydrogenated bisphenol A 本源精化环保科技有限公司 2024-08-16 CN claimed
CN-118459369-A Synthetic method of N-Boc-vinyl glycine methyl ester and isomer thereof 成都师范学院 2024-08-09 CN claimed
CN-118398109-A Physical property data prediction method and device for flow simulation 广东辛孚科技有限公司 2024-07-26 CN claimed
EP-0924521-A1 Competitive apo-peroxidase assay Bayer Corporation (US) 1999-06-23 EP claimed
CN-1210856-A Process for preparation of heteroarylcarboxamides AMERICAN CYANAMID CO (US) 1999-03-17 CN claimed
CN-1041513-C Inhibiting polymerization of vinyl aromatic monomers CIBA GEIGY AG (CH) 1999-01-06 CN claimed
EP-0882700-A2 Process for the production of the dexfenfluramine hydrochloride ALFA CHEMICALS ITALIANA S.p.A. (IT) 1998-12-09 EP claimed
CN-1185209-A Assaying protein fragments in body fluids OSTEOMETER BIOTECH AS (DK) 1998-06-17 CN claimed
CN-1166820-A Method for inhibiting premature polymerization of aromatic vinyl monomers CIBA GEIGY AG (CH) 1997-12-03 CN claimed
CN-1163312-A Novel sphingomyelin and its preparing method ROHM & HAAS (US) 1997-10-29 CN claimed
CN-1121202-A Chinese character input method for computer LIU LIANXUN (CN) 1996-04-24 CN claimed
CN-1084155-A The resistance of vi-ny l aromatic monomers is poly- CIBA GEIGY AG (US) 1994-03-23 CN claimed
CN-1053859-A Reclaim the method for the plutonium (IV) in solution such as waste water, fission product strong solution and the concentrated solution of plutonium with crown compound COGEMA COMPAGNIC GENERALE DES (FR) 1991-08-14 CN claimed