SCHEMBL12100962

SCHEMBL12100962

Cc1nc(C(=O)N2CCCC3(CCN(CCCCCCCCC=O)CC3)C2)cs1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.43
CHRM3 P20309 3/20 0.43
CYP3A4 P08684 15/20 0.43
CYP2D6 P10635 12/20 0.43
USP2 O75604 3/20 0.43
HSD17B10 Q99714 1/20 0.42
TSHR P16473 5/20 0.40
CYP2C19 P33261 4/20 0.40
ALDH1A1 P00352 3/20 0.39
CYP1A2 P05177 3/20 0.39
CYP2C9 P11712 3/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2141841 0.83 CHRM2 (0.64) CHRM2CHRM3
SCHEMBL12095659 0.81 CHRM2 (0.58) CHRM2CHRM3CYP3A4CYP2D6USP2
SCHEMBL12101048 0.74 CYP3A4 (0.49) CYP3A4CYP2D6USP2HSD17B10TSHR
SCHEMBL2142020 0.72 CHRM2 (0.67) CHRM2CHRM3
SCHEMBL12101073 0.70 CHRM2 (0.45) CHRM2CHRM3CYP3A4CYP2D6USP2
SCHEMBL29944255 0.68 NPC1 (0.57) HSD17B10TSHRALDH1A1MEN1KMT2A
SCHEMBL12101040 0.67 GRM5 (0.43) CYP3A4CYP2D6USP2TSHRCYP2C19
SCHEMBL12101012 0.65 CHRM2 (0.56) CHRM2CHRM3CYP3A4CYP2D6USP2
SCHEMBL2142054 0.65 CHRM2 (0.63) CHRM2CHRM3
SCHEMBL19107352 0.65 CHRM2 (0.61) CHRM2CHRM3ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2242759-B1 COMPOUNDS ASTRAZENECA AB (SE) 2012-09-12 EP disclosed