SCHEMBL12101040

SCHEMBL12101040

Cc1ccc(C(=O)N2CCCC3(CCN(CCCCCCCCCO)CC3)C2)s1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.43
SLC6A1 P30531 1/20 0.42
HRH2 P25021 1/20 0.41
HRH1 P35367 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 14/20 0.40
CYP2D6 P10635 11/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 1/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
TSHR P16473 2/20 0.38
USP2 O75604 2/20 0.38
HTR1A P08908 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2140502 0.82 CHRM2 (0.46) HRH2HRH1
SCHEMBL12101084 0.79 CYP3A4 (0.43) GRM5CYP3A4CYP2D6ALDH1A1CYP1A2
SCHEMBL12100972 0.79 CYP3A4 (0.46) GRM5CYP3A4CYP2D6ALDH1A1HPGD
SCHEMBL12100975 0.76 CYP3A4 (0.40) GRM5POLBCYP3A4CYP2D6ALDH1A1
SCHEMBL12100964 0.75 CYP3A4 (0.46) GRM5CYP3A4CYP2D6ALDH1A1HPGD
SCHEMBL4379805 0.72 SLC6A1 (0.38) GRM5SLC6A1POLBCYP3A4CYP2D6
SCHEMBL12101048 0.72 CYP3A4 (0.49) GRM5CYP3A4CYP2D6ALDH1A1CYP1A2
SCHEMBL16132007 0.72 ALDH1A1 (0.56) HRH2HRH1POLBALDH1A1HPGD
SCHEMBL4157157 0.69 HPGD (0.66) POLBALDH1A1HPGD
SCHEMBL17319591 0.69 HPGD (0.66) POLBALDH1A1HPGDHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2242759-B1 COMPOUNDS ASTRAZENECA AB (SE) 2012-09-12 EP disclosed