SCHEMBL12101048

SCHEMBL12101048

O=C(c1csc(-c2ccccc2)n1)N1CCCC2(CCN(CCCCCCCCCO)CC2)C1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 13/20 0.49
CYP2D6 P10635 8/20 0.49
USP2 O75604 5/20 0.49
TSHR P16473 3/20 0.49
ACKR3 P25106 2/20 0.45
CYP1A2 P05177 7/20 0.42
CYP2C19 P33261 5/20 0.42
ALDH1A1 P00352 3/20 0.42
CYP2C9 P11712 3/20 0.42
HSD17B10 Q99714 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
GRM5 P41594 1/20 0.42
PIN1 Q13526 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2139692 0.84 CHRM2 (0.58) ACKR3PTGDR2
SCHEMBL12101047 0.76 ADRB2 (0.39) CYP3A4CYP2D6USP2TSHR
SCHEMBL12100962 0.74 CHRM2 (0.43) CYP3A4CYP2D6USP2TSHRCYP1A2
SCHEMBL29944217 0.73 HTR2C (0.63) ALDH1A1HSD17B10PTGDR2MEN1KMT2A
SCHEMBL3547467 0.73 HTR2C (0.63) ALDH1A1HSD17B10PTGDR2MEN1KMT2A
SCHEMBL3543198 0.73 HTR2C (0.63) ALDH1A1HSD17B10PTGDR2MEN1KMT2A
SCHEMBL12101040 0.72 GRM5 (0.43) CYP3A4CYP2D6USP2TSHRCYP1A2
SCHEMBL12101045 0.70 CYP3A4 (0.39) CYP3A4CYP2D6USP2TSHRCYP1A2
SCHEMBL12101084 0.69 CYP3A4 (0.43) CYP3A4CYP2D6USP2TSHRCYP1A2
SCHEMBL12101088 0.69 CHRM2 (0.43) CYP3A4CYP2D6USP2TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2242759-B1 COMPOUNDS ASTRAZENECA AB (SE) 2012-09-12 EP disclosed