SCHEMBL12101047

SCHEMBL12101047

CN(CCCCCCCCCN1CCC2(CCCN(C(=O)c3csc(-c4ccccc4)n3)C2)CC1)C[C@H](O)c1ccc(O)c2[nH]c(=O)sc12

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 19/20 0.39
ADRB1 P08588 13/20 0.39
DRD2 P14416 3/20 0.39
USP2 O75604 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
ADRA1D P25100 1/20 0.35
CHRM3 P20309 1/20 0.34
DRD3 P35462 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10242601 0.78 ADRB2 (0.52) ADRB2ADRB1DRD2ADRA1DCHRM3
SCHEMBL12101076 0.78 ADRB2 (0.47) ADRB2ADRB1DRD2ADRA1DCHRM3
Formic Acid SCHEMBL2142847 0.77 ADRB2 (0.51) ADRB2ADRB1DRD2ADRA1DCHRM3
Formic Acid SCHEMBL2142822 0.77 ADRB2 (0.51) ADRB2ADRB1DRD2ADRA1DCHRM3
SCHEMBL12101048 0.76 CYP3A4 (0.49) USP2CYP3A4CYP2D6TSHR
SCHEMBL12100968 0.74 ADRB2 (0.55) ADRB2ADRB1DRD2ADRA1DCHRM3
SCHEMBL2139288 0.74 CHRM3 (0.44) ADRB2ADRB1CHRM3DRD3
SCHEMBL2142827 0.73 ADRB2 (0.44) ADRB2ADRB1DRD2CHRM3
SCHEMBL12100965 0.72 ADRB2 (0.47) ADRB2ADRB1DRD2ADRA1DCHRM3
SCHEMBL2140483 0.72 CHRM3 (0.42) ADRB2ADRB1DRD2ADRA1DCHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2242759-B1 COMPOUNDS ASTRAZENECA AB (SE) 2012-09-12 EP disclosed