Alpha-Naphthoflavone

Alpha-Naphthoflavone

SCHEMBL121594

O=c1cc(-c2ccccc2)oc2c1ccc1ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 14/20 1.00
CYP1B1 Q16678 14/20 1.00
CYP1A2 P05177 13/20 1.00
PRKDC P78527 4/20 1.00
CYP19A1 P11511 2/20 1.00
KDM4E B2RXH2 2/20 1.00
ABCB1 P08183 2/20 1.00
ABCC1 P33527 2/20 1.00
ABCG2 Q9UNQ0 2/20 1.00
PDE5A O76074 1/20 1.00
ALDH1A1 P00352 1/20 1.00
TP53 P04637 1/20 1.00
CYP3A4 P08684 1/20 1.00
CYP2D6 P10635 1/20 1.00
MAPT P10636 1/20 1.00
CYP2C9 P11712 1/20 1.00
HPGD P15428 1/20 1.00
TSHR P16473 1/20 1.00
CYP2B6 P20813 1/20 1.00
TACR2 P21452 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alpha-Naphthoflavone SCHEMBL29351090 1.00 CYP1A1 (1.00) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1
Alpha-Naphthoflavone SCHEMBL17292887 0.92 CYP1A1 (0.84) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1
Alpha-Naphthoflavone SCHEMBL3665037 0.90 CYP1A1 (0.82) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1
Alpha-Naphthoflavone SCHEMBL1906540 0.89 CYP1A1 (0.80) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1
SCHEMBL4069839 0.88 CYP1A1 (1.00) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1
SCHEMBL20594586 0.88 CYP1A1 (0.78) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1
SCHEMBL29407618 0.88 CYP1A1 (0.78) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1
SCHEMBL30917246 0.88 CYP1A1 (1.00) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1
SCHEMBL31061133 0.88 PRKDC (1.00) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1
SCHEMBL31061033 0.86 CYP1A1 (1.00) CYP1A1CYP1B1CYP1A2PRKDCCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2073 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119138363-A Method for creating golden pomfret pseudo-male fish 海南大学三亚南繁研究院 2024-12-17 CN claimed
CN-118661742-A Insecticidal composition and application thereof in loquat pest control 四川农业大学 2024-09-20 CN claimed
US-20240269066-A1 USE OF CYP450 INHIBITOR IN INHIBITING OR KILLING MITES AND TREATING XEROPHTHALMIA PRECVISION BIOTECHNOLOGIES LTD. (CN) 2024-08-15 US claimed
EP-4353264-A1 USE OF CYP450 INHIBITOR IN INHIBITING OR KILLING MITES AND TREATING DRY EYE SYNDROME Precvision Biotechnologies Ltd. (CN) 2024-04-17 EP claimed
CN-117897141-A Flavonoid-rich spray-dried powder 梅西大学 2024-04-16 CN claimed
EP-4284386-A1 FLAVONOID-ENRICHED SPRAY-DRIED POWDER Massey University (NZ) 2023-12-06 EP claimed
US-20230126434-A1 OPTIMIZED CRISPR/CAS9 SYSTEMS AND METHODS FOR GENE EDITING IN STEM CELLS EDITAS MEDICINE, INC. 2023-04-27 US claimed
EP-3524604-B1 EXPANDED HEMATOPOIETIC STEM CELLS FROM CORD BLOOD AND THEIR THERAPEUTIC USE NOVARTIS AG (CH) 2023-03-29 EP claimed
US-20230032216-A1 INTERLEUKIN-4-INDUCED GENE 1 (IL4I1) AND RESPECTIVE METABOLITES AS BIOMARKERS FOR CANCER Deutsches Krebsforschungszentrum Stiftung des oeffentlichen Rechts Im Neuenheimer Feld 280 (DE) 2023-02-02 US claimed
WO-2022257986-A1 USE OF CYP450 INHIBITOR IN INHIBITING OR KILLING MITES AND TREATING DRY EYE SYNDROME 广州岐微生物医药科技有限公司 2022-12-15 WO claimed
US-6066642-A FOR SELECTIVELY BLOCKING THE A3 ADENOSINE RECEPTOR OF A MAMMAL THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-05-23 US claimed
EP-0985166-A1 METHODS OF IMAGING AND PRINTING WITH A POSITIVE-WORKING INFRARED RADIATION SENSITIVE PRINTING PLATE Kodak Polychrome Graphics LLC (US) 2000-03-15 EP claimed
EP-0954304-A2 METHODS FOR REGULATING NICOTINE METABOLISM Nicogen Inc. (CA) 1999-11-10 EP claimed
US-5886157-A EXTRACTING THE PROTEIN FROM MEMBRANE CELLS WITH NONIONIC DETERGENT, CENTRIFUGING, PURIFYING THROUGH CHROMATOGRAPHIC COLUMN VANDERBILT UNIVERSITY (US) 1999-03-23 US claimed
WO-1999007381-A1 COMPOSITIONS AND TREATMENTS TO REDUCE SIDE EFFECTS OF ADMINISTRATION OF ANDROGENIC TESTOSTERONE PRECURSORS WEIDER NUTRITION INTERNATIONAL, INC. (US) 1999-02-18 WO claimed
WO-1998054621-A1 METHODS OF IMAGING AND PRINTING WITH A POSITIVE-WORKING INFRARED RADIATION SENSITIVE PRINTING PLATE KODAK POLYCHROME GRAPHICS, L.L.C. (US) 1998-12-03 WO claimed
WO-1998003171-A2 USE OF INHIBITORS OF CYP2A6 FOR REGULATING NICOTINE METABOLISM NICOGEN INC. (CA) 1998-01-29 WO claimed
US-5663029-A DEVELOPMENT OF LATENT IMAGE, TRANSFERRING TO FORM RECORDING SHEETS, COATING A SUBSTRATE USING POLYMERS XEROX CORPORATION (US) 1997-09-02 US claimed
WO-1994023715-A1 USE OF FLAVONOIDS TO TREAT MULTIDRUG RESISTANT CANCER CELLS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-10-27 WO claimed
US-5336685-A Use of flavonoids to treat multidrug resistant cancer cells SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-08-09 US claimed