SCHEMBL12178754

SCHEMBL12178754

OC1(c2nccs2)CC2CCCNC2C1

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.34
NR3C1 P04150 1/20 0.31
ADORA2A P29274 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12178707 0.76 SMN1; SMN2 (0.32)
SCHEMBL30479589 0.75 OPRL1 (0.40) OPRL1NR3C1
SCHEMBL12178738 0.74 CHRNB2 (0.35)
SCHEMBL12179332 0.73 CHRNB2 (0.33)
SCHEMBL12179327 0.73 CHRM2 (0.38) OPRL1
SCHEMBL2584526 0.72 OPRL1 (0.40) OPRL1NR3C1
SCHEMBL12179170 0.72 OPRM1 (0.36) OPRL1
SCHEMBL12178751 0.71 CHRM2 (0.44)
SCHEMBL15825000 0.70 OPRL1 (0.39) OPRL1
SCHEMBL12178857 0.70 CHRNB2 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011135276-A1 3, 3 -DISUBSTITUTED- ( 8 - AZA - BICYCLO [3.2.1] OCT- 8 - YL) -[5- (1H - PYRAZOL - 4 -YL) -THIOPHEN-3 -YL] METHANONES AS INHIBITORS OF 11 (BETA) -HSD1 THE UNIVERSITY OF EDINBURGH (GB) 2011-11-03 WO disclosed