SCHEMBL12195705

SCHEMBL12195705

C=C(NCc1ccccc1)C1(c2ccccc2)CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.51
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
CYP2C19 P33261 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
HDAC1 Q13547 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
HDAC3 O15379 1/20 0.48
HDAC2 Q92769 1/20 0.48
OPRD1 P41143 1/20 0.48
OPRK1 P41145 1/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA7 P43166 2/20 0.48
CA9 Q16790 2/20 0.48
HTT P42858 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KDM1A O60341 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2468207 0.88 ALDH1A1 (0.60) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL13182885 0.87 GRIN2B (0.54) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL2470472 0.84 OPRL1 (0.56) SMN1; SMN2NPC1RAB9AMEN1KMT2A
SCHEMBL2467789 0.83 KMT2A (0.58) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL2493540 0.81 TACR1 (0.53) MEN1KMT2ANPSR1HDAC1HDAC6
SCHEMBL16639868 0.81 SMN1; SMN2 (0.59) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL3901930 0.81 OPRD1 (0.56) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL6759957 0.81 HDAC1 (0.57) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL2498809 0.80 ALDH1A1 (0.59) SMN1; SMN2CYP2C19MEN1KMT2ANPSR1
SCHEMBL4631143 0.80 OPRD1 (0.53) SMN1; SMN2NPC1RAB9ACYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2371366-A1 Heterocyclo inhibitors of potassium channel function Bristol-Myers Squibb Company (US) 2011-10-05 EP disclosed
EP-2228065-A2 Heterocyclo inhibitors of potassium channel function Bristol-Myers Squibb Company (US) 2010-09-15 EP disclosed