SCHEMBL12197814

SCHEMBL12197814

C=C1c2cc(N)c(C)cc2OCN1C1CC1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12197818 0.75 CYP19A1 (0.36)
SCHEMBL8081279 0.64 CYP3A4 (0.37) CYP3A4TSHRMAPK1
SCHEMBL4070655 0.62 ALDH1A1 (0.37) CYP3A4TSHR
SCHEMBL4067017 0.61 CYP19A1 (0.41)
SCHEMBL29362737 0.61 ALDH1A1 (0.47) CYP3A4TSHRMAPK1
SCHEMBL30030734 0.61 MEN1 (0.47) CYP3A4TSHRMAPK1
SCHEMBL1027495 0.61 MEN1 (0.47) CYP3A4TSHRMAPK1
SCHEMBL3344312 0.61 ALDH1A1 (0.47) CYP3A4TSHRMAPK1
SCHEMBL2789554 0.59 AR (0.45)
SCHEMBL16253981 0.57 MAPT (0.51) CYP3A4TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144506-B1 3-SUBSTITUTED-[1,2,3]-BENZOTRIAZINONE COMPOUND FOR ENHANCING GLUTAMATERGIC SYNAPTIC RESPONSES CORTEX PHARMA INC (US) 2011-10-05 EP disclosed