SCHEMBL12199033

SCHEMBL12199033

COC(=O)[C@@H](C)Cc1c[nH]cn1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.33
THRB P10828 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ESRRB O95718 1/20 0.32
DYRK1A Q13627 1/20 0.32
MAP3K7 O43318 2/20 0.31
TAB1 Q15750 2/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
BAZ2B Q9UIF8 1/20 0.31
BAZ2A Q9UIF9 1/20 0.31
MAPK1 P28482 1/20 0.31
HDAC6 Q9UBN7 4/20 0.30
HDAC1 Q13547 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10276525 1.00 ALDH1A1 (0.35) ALDH1A1SMN1; SMN2THRBCYP2C9CYP2C19
SCHEMBL21782663 0.86 MEN1 (0.33) ALDH1A1SMN1; SMN2
SCHEMBL21266611 0.85 CYP1A2 (0.37) CYP2C9ESR1ESR2
SCHEMBL23048409 0.85 NLRP3 (0.32) ALDH1A1MAP3K7TAB1
SCHEMBL16452416 0.84 SMN1; SMN2 (0.31) ALDH1A1SMN1; SMN2MAP3K7TAB1
SCHEMBL16452417 0.84 SMN1; SMN2 (0.31) ALDH1A1SMN1; SMN2MAP3K7TAB1
SCHEMBL833709 0.84 ALDH1A1 (0.36) ALDH1A1MAP3K7TAB1
SCHEMBL8365459 0.84 ESR1 (0.33) ESR1ESR2
SCHEMBL262238 0.84 ALDH1A1 (0.36) ALDH1A1MAP3K7TAB1
SCHEMBL29103272 0.84 HDAC6 (0.36) ALDH1A1THRBCYP2C9CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2371421-A1 Ligands of insulin degrading enzyme and their uses Université de Lille 2 Droit et Santé (FR) 2011-10-05 EP disclosed
WO-2011107948-A2 LIGANDS OF INSULIN DEGRADING ENZYME AND THEIR USES UNIVERSITE LILLE 2 DROIT ET SANTE (FR) 2011-09-09 WO disclosed