SCHEMBL12200056

SCHEMBL12200056

CCc1cc2c(cc1CC)[C@H](CCc1ccc(C(F)(F)F)cc1)NCC2

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.45
TBXA2R P21731 1/20 0.45
KDM1A O60341 5/20 0.44
GAA P10253 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
DRD2 P14416 2/20 0.38
DRD4 P21917 2/20 0.38
MEN1 O00255 1/20 0.38
ABL1 P00519 1/20 0.38
ALPL P05186 1/20 0.38
KMT2A Q03164 1/20 0.38
RIN1 Q13671 1/20 0.38
SLC6A3 Q01959 1/20 0.37
BCHE P06276 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12200036 0.89 BCHE (0.47) GAAKDM4EMAPTHTTKMT2A
SCHEMBL1680336 0.83 BCHE (0.57) KDM4EMAPTKMT2ABCHE
SCHEMBL3346743 0.83 BCHE (0.57) KDM4EMAPTKMT2ABCHE
SCHEMBL990798 0.83 BCHE (0.57) KDM4EMAPTKMT2ABCHE
Hydrochloric Acid SCHEMBL987382 0.82 BCHE (0.56) KDM4EMAPTKMT2ABCHE
Acetic Acid SCHEMBL3169809 0.80 MTNR1B (0.54) KDM4EMAPTKMT2ABCHE
Acetic Acid SCHEMBL990742 0.80 MTNR1B (0.54) KDM4EMAPTKMT2ABCHE
Hydrochloric Acid SCHEMBL3654652 0.79 BCHE (0.47) ADRB2TBXA2RGAAKDM4EMAPT
SCHEMBL1364512 0.74 L3MBTL1 (0.41) ADRB2TBXA2RKDM1A
SCHEMBL1364766 0.72 L3MBTL1 (0.43) ADRB2TBXA2RKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2227455-B1 TRISUBSTITUTED 3,4-DIHYDRO-1H-ISOQUINOLIN COMPOUND, PROCESS FOR ITS PREPARATION, AND ITS USE ACTELION PHARMACEUTICALS LTD (CH) 2011-10-12 EP disclosed