SCHEMBL12205342

SCHEMBL12205342

CC(C)(C)OC(=O)CN1C(=O)C2(CC(=O)NC2=O)c2cc(N)ccc21

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 10/20 0.37
AKR1B1 P15121 2/20 0.34
NR1H2 P55055 1/20 0.34
OPRL1 P41146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2480752 0.88 PTGDR2 (0.51) PTGDR2AKR1B1
SCHEMBL11959139 0.76 PTGDR2 (0.54) PTGDR2AKR1B1
SCHEMBL11959133 0.75 PTGDR2 (0.48) PTGDR2
SCHEMBL4394762 0.70 PTGDR2 (0.67) PTGDR2
SCHEMBL4958492 0.69 PTGDR2 (0.46) PTGDR2
SCHEMBL11959132 0.69 PTGDR2 (0.44) PTGDR2OPRL1
SCHEMBL2483141 0.69 PTGDR2 (0.75) PTGDR2
SCHEMBL5007572 0.67 ALDH1A1 (0.46) OPRL1
SCHEMBL14876503 0.67 CASP1 (0.52)
SCHEMBL22040148 0.66 NR1H2 (0.35) NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891075-B1 TRICYCLIC SPIRO DERIVATIVES AS CRTH2 MODULATORS MERCK SERONO SA (CH) 2011-10-19 EP disclosed