SCHEMBL12207

SCHEMBL12207

C=C1N(c2ccc(C(C)(C)C)cc2)CC[C@]12CC[C@@](O)(CC)CC2

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 10/20 0.40
TRPV1 Q8NER1 1/20 0.35
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
KCNH2 Q12809 1/20 0.32
HSD11B1 P28845 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12342 0.82 LIPE (0.52) LIPETRPV1DRD2KCNH2
SCHEMBL12336 0.81 TRPV1 (0.33) LIPETRPV1DRD2DRD3KCNH2
SCHEMBL10019 0.75 LIPE (0.69) LIPETRPV1
SCHEMBL10020 0.75 LIPE (0.69) LIPETRPV1
SCHEMBL5706 0.72 LIPE (0.55) LIPETRPV1
SCHEMBL5705 0.72 LIPE (0.55) LIPETRPV1
SCHEMBL12702552 0.72 LIPE (0.55) LIPETRPV1
SCHEMBL1589386 0.72 LIPE (0.53) LIPETRPV1
SCHEMBL1589384 0.72 LIPE (0.53) LIPETRPV1
SCHEMBL12702141 0.72 LIPE (0.53) LIPE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011045292-A1 SPIRO-CONDENSED CYCLOHEXANE DERIVATIVES AS HSL INHIBITORS USEFUL FOR THE TREATMENT OF DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2011-04-21 WO disclosed