SCHEMBL12336

SCHEMBL12336

C=C1N(c2ccc(C(C)(C)C)cc2)CC[C@]12CC[C@@](C)(C(O)CC)CC2

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.33
LIPE Q05469 3/20 0.32
MAPT P10636 1/20 0.31
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12207 0.81 LIPE (0.40) TRPV1LIPEDRD2DRD3KCNH2
SCHEMBL12342 0.72 LIPE (0.52) TRPV1LIPEDRD2KCNH2
SCHEMBL1589896 0.68 EBP (0.44) TRPV1LIPE
SCHEMBL12702580 0.68 EBP (0.44) TRPV1LIPE
SCHEMBL1589897 0.68 EBP (0.44) TRPV1LIPE
SCHEMBL10019 0.65 LIPE (0.69) TRPV1LIPE
SCHEMBL10020 0.65 LIPE (0.69) TRPV1LIPE
SCHEMBL9814 0.64 LIPE (0.46) TRPV1LIPE
SCHEMBL9815 0.64 LIPE (0.46) TRPV1LIPE
SCHEMBL12443370 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011045292-A1 SPIRO-CONDENSED CYCLOHEXANE DERIVATIVES AS HSL INHIBITORS USEFUL FOR THE TREATMENT OF DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2011-04-21 WO disclosed