SCHEMBL12207656

SCHEMBL12207656

CC1(C)C(=O)N(Cc2ccsc2)c2cc3[nH]c(N)nc3cc21

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
PNP P00491 5/20 0.37
RAF1 P04049 1/20 0.34
BRAF P15056 1/20 0.34
FABP6 P51161 1/20 0.33
ALDH1A1 P00352 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TYMS P04818 10/20 0.31
DHFR P00374 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2490810 0.82 AURKA (0.40) AURKAAURKBRAF1BRAFFABP6
SCHEMBL13367949 0.78 AURKA (0.47) AURKAAURKBRAF1BRAFFABP6
SCHEMBL2491924 0.78 AURKA (0.45) AURKAAURKBRAF1BRAFFABP6
SCHEMBL2488865 0.78 AURKA (0.42) AURKAAURKBRAF1BRAFFABP6
SCHEMBL2490394 0.76 AURKA (0.42) AURKAAURKBRAF1BRAFFABP6
SCHEMBL10693758 0.76 AURKA (0.41) AURKAAURKBPNPALDH1A1
SCHEMBL2487407 0.76 AURKA (0.64) AURKAAURKBRAF1BRAFFABP6
SCHEMBL3424973 0.74 AURKA (0.44) AURKAAURKBRAF1BRAFFABP6
SCHEMBL2489572 0.74 AURKA (0.37) AURKAAURKBTYMS
SCHEMBL2491051 0.74 AURKA (0.41) AURKAAURKBFABP6ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756112-B1 PYRROLOBENZIMIDAZOLONES AND THEIR USE AS ANTIPROLIFERATIVE AGENTS BOEHRINGER INGELHEIM INT (DE) 2011-10-26 EP disclosed