SCHEMBL10693758

SCHEMBL10693758

CCCCN1C(=O)C(C)(C)c2cc3nc(Cc4ccsc4)[nH]c3cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.41
AURKB Q96GD4 2/20 0.41
PNP P00491 2/20 0.35
PABPC1 P11940 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
KDM4A O75164 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
IDH1 O75874 1/20 0.33
KDM4E B2RXH2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KMT2A Q03164 4/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10695723 0.83 LMNA (0.44) AURKAAURKBPNPALDH1A1HPGD
SCHEMBL10695197 0.80 AURKA (0.46) AURKAAURKBALDH1A1HPGDKDM4A
SCHEMBL13341286 0.79 AURKA (0.41) AURKAAURKBSMN1; SMN2KMT2AMEN1
SCHEMBL10696394 0.76 PDE4A (0.52) AURKAAURKBALDH1A1HPGDHSD17B10
SCHEMBL12207656 0.76 AURKA (0.40) AURKAAURKBPNPALDH1A1
SCHEMBL10695665 0.75 RIPK1 (0.48) AURKAAURKBTSHRKDM4ESMN1; SMN2
SCHEMBL13341645 0.75 LMNA (0.40) AURKAAURKBALDH1A1TSHRMAPK1
SCHEMBL2488149 0.74 AURKA (0.48) AURKAAURKBALDH1A1KDM4ESMN1; SMN2
SCHEMBL2485583 0.74 AURKA (0.48) AURKAAURKBHPGDSMN1; SMN2KMT2A
SCHEMBL2486921 0.74 AURKA (0.48) AURKAAURKBNPSR1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed