Benzamide

Benzamide

SCHEMBL1222101

NC(=O)c1ccccc1.NC(=O)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 1.00
TSHR P16473 2/20 1.00
POLB P06746 1/20 1.00
CYP3A4 P08684 1/20 1.00
MAPT P10636 1/20 1.00
CYP2C19 P33261 1/20 1.00
RECQL P46063 1/20 1.00
BLM P54132 1/20 1.00
PMP22 Q01453 1/20 1.00
HSD17B10 Q99714 1/20 1.00
TDP1 Q9NUW8 1/20 1.00
L3MBTL1 Q9Y468 1/20 1.00
PARP10 Q53GL7 4/20 0.62
PLA2G10 O15496 1/20 0.62
PLA2G2A P14555 1/20 0.62
CES2 O00748 2/20 0.58
CES1 P23141 2/20 0.58
ALDH1A1 P00352 2/20 0.58
DAO P14920 1/20 0.58
NAPRT Q6XQN6 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21755166 1.00 PARP1 (1.00) PARP1TSHRPOLBCYP3A4MAPT
Benzamide SCHEMBL30112947 1.00 PARP1 (1.00) PARP1TSHRPOLBCYP3A4MAPT
Benzamide SCHEMBL11668921 1.00 PARP1 (1.00) PARP1TSHRPOLBCYP3A4MAPT
Benzamide SCHEMBL6690447 1.00 PARP1 (1.00) PARP1TSHRPOLBCYP3A4MAPT
Benzamide SCHEMBL16352 1.00
Benzamide SCHEMBL27963599 1.00 PARP1 (1.00) PARP1TSHRPOLBCYP3A4MAPT
Benzamide SCHEMBL29618402 1.00
Benzamide SCHEMBL1332331 1.00
Benzamide SCHEMBL8961640 0.97 PARP1 (0.94) PARP1TSHRPOLBCYP3A4MAPT
Benzamide SCHEMBL3864950 0.97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3227272-A1 BIFUNCTIONAL do2pa DERIVATIVES, CHELATES WITH METALLIC CATIONS AND USE THEREOF Centre National de la Recherche Scientifique (CNRS) (FR) 2017-10-11 EP disclosed
CN-103819459-B Anti-Viral Compounds 艾伯维巴哈马有限公司 2017-05-17 CN disclosed
CN-106573929-A 1h-1,8- naphthyridin-2ones as anti proliferative compounds 纳科法尔马有限公司 2017-04-19 CN disclosed
WO-2016087667-A1 BIFUNCTIONAL do2pa DERIVATIVES, CHELATES WITH METALLIC CATIONS AND USE THEREOF CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2016-06-09 WO disclosed
CN-103172620-B Anti-viral compounds Abbott Labaoratories (BS) 2014-10-29 CN disclosed
CN-103819459-A Anti-Viral Compounds Abbott Labaoratories 2014-05-28 CN disclosed
CN-103819537-A Anti-viral compounds Abbott Labaoratories 2014-05-28 CN disclosed
CN-102333772-B Antiviral compounds ABBOTT LAB 2013-12-11 CN disclosed
CN-103172620-A Anti-viral compounds Abbott Labaoratories 2013-06-26 CN disclosed
CN-102333772-A Antiviral compounds ABBOTT LAB 2012-01-25 CN disclosed
CN-1104439-C Phenyl-substituted 4-azasteroid fluoro derivatives, process for their preparation and their use as medicaments PHAMACIA & UPJOHN S P A (IT) 2003-04-02 CN disclosed
CN-1313762-A Apomorphine-containing dosage forms for ameliorating male erectile dysfunction PENTECH PHARMACEUTICALS INC (US) 2001-09-19 CN disclosed
CN-1218399-A Benzamide treatment of dementia associated with AIDs virus (HIV-4) infection CENTAUR PHARMACEUTICALS INC (US) 1999-06-02 CN disclosed
CN-1165520-A Phenylsubstituted 4-azasteroid fluoroderivatives PHARMACIA SPA (IT) 1997-11-19 CN disclosed
US-5382600-A 3,3-diphenylpropylamines and pharmaceutical compositions thereof PHARMACIA AKTIEBOLAG (SE) 1995-01-17 US disclosed
US-5167876-A Protective clothing; military aircraft interiors ALLIED-SIGNAL INC. (US) 1992-12-01 US disclosed
EP-0325571-B1 NEW AMINES, THEIR USE AND PREPARATION Kabi Pharmacia AB (SE) 1991-08-07 EP disclosed
EP-0354234-A1 NEW AMINES, THEIR USE AND PREPARATION KabiVitrum AB (SE) 1990-02-14 EP disclosed
WO-1989006644-A1 NEW AMINES, THEIR USE AND PREPARATION KABIVITRUM AB (SE) 1989-07-27 WO disclosed
EP-0325571-A1 New amines, their use and preparation Kabi Pharmacia AB (SE) 1989-07-26 EP disclosed