SCHEMBL12228209

SCHEMBL12228209

O[C@H]1CC[C@H](C2CCC(c3cc(F)c(F)c(F)c3)CC2)CC1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.42
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
KCNH2 Q12809 1/20 0.30
CES2 O00748 1/20 0.30
CES1 P23141 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17827799 0.90 CES2 (0.31) CES2CES1
SCHEMBL6456856 0.90 ESR2 (0.34) ESR2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6456852 0.90 ESR2 (0.34) ESR2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8767030 0.84 ALDH1A1 (0.33)
SCHEMBL18458536 0.83 ESR2 (0.47) ESR2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL12997531 0.83 CES2 (0.35) ESR2CES2CES1
SCHEMBL18458823 0.83 ESR2 (0.40) ESR2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL13557300 0.82 ALDH1A1 (0.32)
SCHEMBL19619469 0.82 ESR2 (0.30) ESR2
SCHEMBL8623567 0.81 ESR2 (0.48) ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8043670-B2 Polymerizable mesogenic cyclohexyl derivatives MERCK PATENT GMBH (DE) 2011-10-25 US disclosed
US-8043670-B2 Polymerizable mesogenic cyclohexyl derivatives MERCK PATENT GMBH (DE) 2011-10-25 US disclosed
EP-1626079-B1 Polymerisable mesogenic cyclohexylphenyl derivatives MERCK PATENT GMBH (DE) 2008-04-02 EP disclosed