SCHEMBL12285334

SCHEMBL12285334

COc1ccc2[nH]c(I)cc(=O)c2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.69
HPGD P15428 8/20 0.69
KDM4E B2RXH2 9/20 0.63
SMN1; SMN2 Q16637 4/20 0.63
RAB9A P51151 4/20 0.63
NPC1 O15118 3/20 0.63
MAPT P10636 3/20 0.59
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
HSD17B10 Q99714 2/20 0.59
TSHR P16473 1/20 0.59
GFER P55789 1/20 0.59
LMNA P02545 2/20 0.58
GHSR Q92847 1/20 0.55
ABCG2 Q9UNQ0 1/20 0.54
MAPK1 P28482 1/20 0.53
PKM P14618 1/20 0.52
MCL1 Q07820 1/20 0.52
HKDC1 Q2TB90 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20605617 0.81 ALDH1A1 (1.00) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A
SCHEMBL2465149 0.78 ALDH1A1 (1.00) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A
SCHEMBL9183301 0.78 GHSR (0.71) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A
SCHEMBL12285521 0.77 ABCG2 (0.83) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A
SCHEMBL9452357 0.76 ALDH1A1 (0.63) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A
SCHEMBL3011498 0.76 GHSR (0.65) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A
SCHEMBL19211150 0.76 GHSR (0.65) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A
SCHEMBL13234528 0.76 GHSR (0.65) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A
SCHEMBL2597652 0.76 ALDH1A1 (1.00) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A
SCHEMBL29391519 0.76 ALDH1A1 (1.00) ALDH1A1HPGDKDM4ESMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011127406-A2 ACRIDINES AS INHIBITORS OF HASPIN AND DYRK KINASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2011-10-13 WO disclosed