SCHEMBL12286155

SCHEMBL12286155

c1ccc(-c2[nH]nc3ccccc23)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.52
CYP2C19 P33261 2/20 0.52
NOS1 P29475 1/20 0.52
ALDH1A1 P00352 5/20 0.47
KDM4E B2RXH2 4/20 0.47
GAA P10253 4/20 0.47
HPGD P15428 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
HSD17B10 Q99714 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAPK1 P28482 1/20 0.47
DYRK1B Q9Y463 2/20 0.46
ALPL P05186 1/20 0.45
IDO1 P14902 1/20 0.45
TTK P33981 1/20 0.45
MAPK10 P53779 1/20 0.45
ELANE P08246 1/20 0.44
TGFBR1 P36897 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17196524 0.96 CYP1A2 (0.48) CYP1A2CYP2C19NOS1ALDH1A1KDM4E
SCHEMBL4197111 0.84 ALK (0.53) CYP1A2CYP2C19NOS1DYRK1BALK
SCHEMBL20834652 0.80 RAB9A (0.53) CYP1A2CYP2C19NOS1ALDH1A1KDM4E
SCHEMBL8142848 0.79 AURKA (0.45) ALDH1A1KDM4EGAAHPGDNPSR1
SCHEMBL17692468 0.77 CYP1A2 (0.60) CYP1A2CYP2C19NOS1ALDH1A1KDM4E
SCHEMBL18627081 0.75 CYP1A2 (0.48) CYP1A2CYP2C19NOS1ALDH1A1KDM4E
SCHEMBL12075154 0.75 CYP1A2 (0.48) CYP1A2CYP2C19NOS1ALDH1A1KDM4E
SCHEMBL12075256 0.72 TGFBR1 (0.51) CYP1A2CYP2C19NOS1ALDH1A1KDM4E
SCHEMBL15504124 0.71 ADORA2A (0.55) CYP1A2CYP2C19NOS1ALDH1A1GAA
SCHEMBL20733831 0.71 ALK (0.44) ALDH1A1KDM4EGAAHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017099360-A1 ORGANIC ELECTROLUMINESCENT COMPOUND AND ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2017-06-15 WO disclosed
WO-2014200244-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2014-12-18 WO disclosed
WO-2011132683-A1 BIS-CARBAZOLE DERIVATIVE, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME 出光興産株式会社 (JP) 2011-10-27 WO disclosed