SCHEMBL12288588

SCHEMBL12288588

Bc1ccc2nc(NC3(c4ncccc4F)CCC3)ncc2c1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 14/20 0.34
HDAC1 Q13547 14/20 0.34
HDAC2 Q92769 14/20 0.34
HDAC6 Q9UBN7 14/20 0.34
ROCK2 O75116 1/20 0.32
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14936829 0.87 ROCK2 (0.39) HDAC3HDAC1HDAC2HDAC6ROCK2
SCHEMBL29724760 0.85 NPC1 (0.39) HDAC3HDAC1HDAC2HDAC6ROCK2
SCHEMBL12288593 0.85 NPC1 (0.39) HDAC3HDAC1HDAC2HDAC6ROCK2
SCHEMBL12288591 0.84 VNN1 (0.40) HDAC6
SCHEMBL29724942 0.84 VNN1 (0.40) HDAC6
SCHEMBL19942160 0.82 ROCK2 (0.33) HDAC3HDAC1HDAC2HDAC6ROCK2
SCHEMBL12288592 0.82 ROCK2 (0.40) HDAC3HDAC1HDAC2HDAC6ROCK2
SCHEMBL29724793 0.82 ROCK2 (0.40) HDAC3HDAC1HDAC2HDAC6ROCK2
SCHEMBL14714309 0.78 HDAC6 (0.39) HDAC3HDAC1HDAC2HDAC6
SCHEMBL14937337 0.76 HDAC6 (0.42) HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011133888-A1 CERTAIN AMINO-PYRIMIDINES, COMPOSITIONS THEREOF, AND METHODS FOR THEIR USE CYTOKINETICS, INC. (US) 2011-10-27 WO disclosed