SCHEMBL12294286

SCHEMBL12294286

C[C@@H]1CCCc2ncnc(N)c21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 2/20 0.54
NOS3 P29474 4/20 0.35
NOS1 P29475 4/20 0.35
NOS2 P35228 4/20 0.35
HTT P42858 2/20 0.34
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 1/20 0.34
MAP4K4 O95819 1/20 0.33
ADK P55263 1/20 0.33
LRRK2 Q5S007 1/20 0.32
ADORA2A P29274 3/20 0.32
PI4KA P42356 3/20 0.32
PI4K2B Q8TCG2 3/20 0.32
PI4K2A Q9BTU6 3/20 0.32
PI4KB Q9UBF8 3/20 0.32
ADORA3 P0DMS8 2/20 0.32
ADORA1 P30542 2/20 0.32
HRH2 P25021 2/20 0.32
HRH3 Q9Y5N1 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2738477 0.89 LIMK1 (0.45) LIMK1HTTNPC1ADKLRRK2
SCHEMBL2738580 0.89 LIMK1 (0.45) LIMK1HTTNPC1ADKLRRK2
SCHEMBL30666554 0.79 LIMK1 (0.40) LIMK1HTTPOLBL3MBTL1HRH2
SCHEMBL30667152 0.74 LIMK1 (0.39) LIMK1NOS3NOS1NOS2HTT
SCHEMBL512854 0.73 HRH3 (0.42) LIMK1NOS3NOS1NOS2L3MBTL1
SCHEMBL17690273 0.71 LIMK1 (0.50) LIMK1NOS3NOS1NOS2HRH2
SCHEMBL12323859 0.70 LIMK1 (0.33) LIMK1NOS3NOS1NOS2ADORA2A
SCHEMBL15576293 0.70 LIMK1 (0.33) LIMK1HTTNPC1ADORA2API4KA
SCHEMBL680907 0.68 LIMK1 (0.33) LIMK1
SCHEMBL17771685 0.68 LIMK1 (0.33) LIMK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049501-B1 HYDROXYLATED AND METHOXYLATED CYCLOPENTA [D] PYRIMIDINES AS AKT PROTEIN KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2011-09-14 EP disclosed