Aminorex

Aminorex

SCHEMBL123039

NC1=NCC(c2ccccc2)O1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
TAAR1 Q96RJ0 1/20 0.43
SLC6A3 Q01959 2/20 0.42
RAB9A P51151 1/20 0.42
MEN1 O00255 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HDAC3 O15379 2/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
NCOR2 Q9Y618 2/20 0.39
HDAC8 Q9BY41 1/20 0.39
ATM Q13315 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ADORA3 P0DMS8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aminorex SCHEMBL6803173 0.87 HDAC3 (0.41) TSHRTAAR1SLC6A3RAB9AMEN1
SCHEMBL31158568 0.81 TSHR (0.50) TSHRSLC6A3MEN1CYP2C19KMT2A
SCHEMBL34460861 0.81 TSHR (0.50) TSHRSLC6A3MEN1CYP2C19KMT2A
Clominorex SCHEMBL121090 0.81 TAAR1 (0.46) TAAR1SLC6A3RAB9AATMSMN1; SMN2
SCHEMBL14301430 0.76 TSHR (0.45) TSHRALDH1A1HPGDATMSMN1; SMN2
SCHEMBL2399688 0.76 TSHR (0.45) TSHRALDH1A1HPGDATMSMN1; SMN2
SCHEMBL1548278 0.76 ALDH1A1 (0.54) TSHRKMT2AALDH1A1HPGDATM
SCHEMBL21033513 0.73 TSHR (0.47) TSHRTAAR1SLC6A3RAB9AMEN1
SCHEMBL5395444 0.73 TSHR (0.38) TSHRSLC6A3MEN1CYP2C19KMT2A
Hydrochloric Acid SCHEMBL30845839 0.72 TSHR (0.45) TSHRTAAR1SLC6A3MEN1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2353 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS INC (US) 2025-09-25 US claimed
WO-2023212244-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS, INC. (US) 2023-11-02 WO claimed
EP-3891505-B1 A METHOD FOR MEASURING A CONCENTRATION OF A BIOMARKER/ANALYTE IN BLOOD FROM MAMMALS REDHOTDIAGNOSTICS AB (SE) 2022-11-30 EP claimed
US-20220187304-A1 A Method for Measuring a Concentration of a Biomarker-Analyte In Blood from Mammals REDHOT DIAGNOSTICS AB (SE) 2022-06-16 US claimed
EP-3891505-A1 A METHOD FOR MEASURING A CONCENTRATION OF A BIOMARKER/ANALYTE IN BLOOD FROM MAMMALS REDHOTDIAGNOSTICS AB (SE) 2021-10-13 EP claimed
WO-2020156849-A1 A METHOD FOR MEASURING A CONCENTRATION OF A BIOMARKER/ANALYTE IN BLOOD FROM MAMMALS. REDHOTDIAGNOSTICS AB (SE) 2020-08-06 WO claimed
EP-3687576-A1 USE OF CANNABIDIOL IN COMBINATION WITH 5-HT2B RECEPTOR AGONISTS OR AMPHETAMINS IN THE TREATMENT OF EPILEPSY GW Research Limited (GB) 2020-08-05 EP claimed
US-20200237683-A1 USE OF CANNABIDIOL IN COMBINATION WITH 5-HT2B RECEPTOR AGONISTS OR AMPHETAMINS IN THE TREATMENT OF EPILEPSY JAZZ PHARMACEUTICALS RESEARCH UK LIMITED (GB) 2020-07-30 US claimed
US-20200060997-A1 TARR Receptor Agonists for Sexual Dysfunction JOHN MCCOY 2020-02-27 US claimed
WO-2019064031-A1 USE OF CANNABIDIOL IN COMBINATION WITH 5-HT2B RECEPTOR AGONISTS OR AMPHETAMINS IN THE TREATMENT OF EPILEPSY GW Research Limited (GB) 2019-04-04 WO claimed
EP-0977572-A1 USE OF NK-1 RECEPTOR ANTAGONISTS FOR TREATING EATING DISORDERS MERCK SHARP & DOHME LTD. (GB) 2000-02-09 EP claimed
WO-1999008112-A1 METHODS OF IDENTIFYING BIOLOGICAL AGENT COMPOSITIONS SUPRATEK PHARMA INC. (CA) 1999-02-18 WO claimed
WO-1998047513-A1 USE OF NK-1 RECEPTOR ANTAGONISTS FOR TREATING EATING DISORDERS MERCK SHARP & DOHME LIMITED (GB) 1998-10-29 WO claimed
US-5684018-A Acyloxyisopropyl carbamates as prodrugs for amine drugs MERCK & CO., INC. (US) 1997-11-04 US claimed
EP-0724450-A1 COMPOSITION FOR WEIGHT REDUCTION CONTAINING EPHEDRINE AND A MINERAL SALT OR CHELATE Keown, Wendy J. (US) 1996-08-07 EP claimed
US-5543405-A MIXTURE OF EPHEDRINE AND CHROMIUM PICOLINATE KEOWN WENDY J (US) 1996-08-06 US claimed
WO-1996018605-A1 ACYLOXYISOPROPYL CARBAMATES AS PRODRUGS FOR AMINE DRUGS MERCK & CO., INC. (US) 1996-06-20 WO claimed
WO-1995011034-A1 COMPOSITION FOR WEIGHT REDUCTION CONTAINING EPHEDRINE AND A MINERAL SALT OR CHELATE KEOWN WENDY J (US) 1995-04-27 WO claimed
US-5096712-A METHOD FOR ENHANCING PERFORMANCE SO AS TO IMPROVE VIGOR AND DECREASE FATIGUE, CONFUSION, TENSION, AND ANXIETY INTERNEURON PHARMACEUTICALS, INC. (US) 1992-03-17 US claimed
US-5019594-A Method for decreasing appetite INTERNEURON PHARMACEUTICALS, INC. (US) 1991-05-28 US claimed