SCHEMBL12326815

SCHEMBL12326815

N#Cc1cccc(-c2cc(NC3CCN(COCc4ccc(CO)cc4)CC3)c3cnccc3c2)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 13/20 0.46
GBA1 P04062 1/20 0.38
UGCG Q16739 1/20 0.38
GBA2 Q9HCG7 1/20 0.38
ROCK1 Q13464 7/20 0.37
MCHR1 Q99705 2/20 0.37
GPR6 P46095 1/20 0.36
PRKCZ Q05513 1/20 0.35
PRKD2 Q9BZL6 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
CCR2 P41597 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12326775 0.87 ROCK2 (0.45) ROCK2ROCK1GPR6PRKCZPRKD2
SCHEMBL2422015 0.84 ROCK2 (0.49) ROCK2ROCK1GPR6PRKCZPRKD2
SCHEMBL13087219 0.84 SLC6A7 (0.46) ROCK2GPR6
SCHEMBL12327362 0.82 ROCK2 (0.40) ROCK2ROCK1MCHR1GPR6PRKCZ
SCHEMBL12327341 0.82 ROCK2 (0.45) ROCK2ROCK1MCHR1GPR6PRKCZ
SCHEMBL2427691 0.81 ROCK2 (0.48) ROCK2ROCK1MCHR1GPR6PRKCZ
SCHEMBL2425776 0.81 ROCK2 (0.56) ROCK2GBA1ROCK1JAK2JAK1
SCHEMBL2427707 0.81 ROCK2 (0.49) ROCK2ROCK1GPR6PRKCZPRKD2
SCHEMBL2422828 0.80 ROCK2 (0.48) ROCK2ROCK1MCHR1GPR6PRKCZ
SCHEMBL13087174 0.80 ROCK2 (0.44) ROCK2GPR6PRKCZPRKD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2366699-A1 8-SUBSTITUTED ISOQUINOLINE DERIVATIVE AND USE THEREOF Asahi Kasei Pharma Corporation (JP) 2011-09-21 EP disclosed