SCHEMBL12326820

SCHEMBL12326820

Pc1cc(NC2CCNCC2)c2cnccc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.44
ROCK1 Q13464 2/20 0.44
CDC42BPB Q9Y5S2 1/20 0.44
PRKD1 Q15139 1/20 0.43
BRD4 O60885 3/20 0.43
ATAD2 Q6PL18 3/20 0.43
DYRK1A Q13627 1/20 0.41
IKBKB O14920 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
PRKCZ Q05513 7/20 0.41
PRKD2 Q9BZL6 5/20 0.41
CYP1A2 P05177 2/20 0.41
LATS1 O95835 1/20 0.41
LATS2 Q9NRM7 1/20 0.41
CYP3A4 P08684 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ALOX15 P16050 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15172430 0.81 PRKCZ (0.43) ROCK2ROCK1CDC42BPBPRKD1BRD4
SCHEMBL12327354 0.81 PRKCZ (0.62) ROCK2ROCK1CDC42BPBIKBKBPRKCZ
SCHEMBL13440618 0.80 PRKCZ (0.47) ROCK2ROCK1CDC42BPBPRKD1BRD4
Hydrochloric Acid SCHEMBL23360683 0.80 PRKCZ (0.48) ROCK2ROCK1CDC42BPBBRD4ATAD2
SCHEMBL13440633 0.79 PRKCZ (0.44) ROCK2ROCK1CDC42BPBPRKD1BRD4
SCHEMBL13090107 0.79 PRKCZ (0.44) ROCK2ROCK1CDC42BPBPRKD1BRD4
SCHEMBL15172427 0.79 PRKCZ (0.44) ROCK2ROCK1CDC42BPBPRKD1PRKCZ
Hydrochloric Acid SCHEMBL23360436 0.78 ROCK2 (0.57) ROCK2ROCK1CDC42BPBBRD4ATAD2
Hydrochloric Acid SCHEMBL29862734 0.78 ROCK2 (0.57) ROCK2ROCK1CDC42BPBBRD4ATAD2
SCHEMBL15172382 0.77 BRD4 (0.46) ROCK2ROCK1CDC42BPBBRD4ATAD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2366699-A1 8-SUBSTITUTED ISOQUINOLINE DERIVATIVE AND USE THEREOF Asahi Kasei Pharma Corporation (JP) 2011-09-21 EP disclosed