SCHEMBL12367222

SCHEMBL12367222

CS(=O)(=O)Oc1ccnc2cnc(Cl)cc12

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MET P08581 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
DOT1L Q8TEK3 1/20 0.33
IDO1 P14902 2/20 0.32
ALDH1A1 P00352 1/20 0.32
PDGFRA P16234 2/20 0.32
PDGFRB P09619 1/20 0.32
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32
KDR P35968 1/20 0.32
NFE2L2 Q16236 1/20 0.32
AXL P30530 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2185158 0.82 PDE4A (0.34) LMNASMN1; SMN2METSLC22A12IDO1
SCHEMBL23528183 0.76 PDGFRA (0.56) METPDGFRAPDGFRBKDR
SCHEMBL29206714 0.75 CSNK2A1 (0.35)
SCHEMBL13457873 0.73 TLR8 (0.38) SMN1; SMN2PDGFRAPDGFRBKDR
SCHEMBL30298724 0.73 NCF1 (0.43) SMN1; SMN2SLC22A12
SCHEMBL30227708 0.70 MPO (0.54) METPDGFRAPDGFRBKDR
SCHEMBL23882523 0.70 MPO (0.54) METPDGFRAPDGFRBKDR
SCHEMBL23146986 0.70 AXL (0.42) LMNASMN1; SMN2IDO1ALDH1A1AXL
SCHEMBL23882454 0.70 FGFR2 (0.43) PDGFRAPDGFRBKDR
SCHEMBL15743523 0.70 PLAU (0.41) LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8735424-B2 Bicyclic kinase inhibitors NOVARTIS AG (CH) 2014-05-27 US disclosed
US-20110195980-A1 Bicyclic Kinase Inhibitors NOVARTIS AG (CH) 2011-08-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110195980-A1 Bicyclic Kinase Inhibitors PIM1, PIM2, PIM3 LMNA 2217/4885SMN1; SMN2 1444/4885MET 1105/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.