SCHEMBL12373214

SCHEMBL12373214

COc1cc(C(C)Cc2ccccc2)c(CO)cc1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 4/20 0.47
CYP3A4 P08684 3/20 0.47
KDM4E B2RXH2 3/20 0.47
GAA P10253 2/20 0.47
TSHR P16473 1/20 0.47
RAB9A P51151 1/20 0.47
ALOX12 P18054 2/20 0.42
FOS P01100 1/20 0.42
TTR P02766 1/20 0.42
JUN P05412 1/20 0.42
NR3C1 P04150 1/20 0.42
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
ATM Q13315 1/20 0.41
MMP1 P03956 1/20 0.40
PTPN7 P35236 1/20 0.40
DUSP3 P51452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1494089 0.90 HTR2A (0.44) ALOX15CYP3A4KDM4EGAATSHR
SCHEMBL5525796 0.84 HTR2A (0.41) ALOX15CYP3A4KDM4EGAATSHR
SCHEMBL5782581 0.81 HTR2A (0.40) ALOX15CYP3A4KDM4EGAATSHR
SCHEMBL16918764 0.75 KDM4E (0.50) ALOX15CYP3A4KDM4EGAATSHR
SCHEMBL5567608 0.74 KMT2A (0.42) RAB9ACYP2D6CYP2C19MAPTMEN1
SCHEMBL20910420 0.73 CYP2D6 (0.68) ALOX15CYP3A4KDM4EGAATSHR
SCHEMBL18065576 0.71 POLB (0.45) ALOX15CYP3A4KDM4EGAATSHR
SCHEMBL1494085 0.70 KDM4E (0.48) ALOX15CYP3A4KDM4EGAATSHR
Mesodihydroguaiaretic Acid SCHEMBL4852003 0.70 FOS (0.84) ALOX15CYP3A4KDM4EGAATSHR
SCHEMBL1494045 0.69 ALDH1A1 (0.45) ALOX15CYP3A4KDM4EGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8008313-B2 Methods of using diaminopyrimidine P2X3 and P2X2/3 receptor modulators for treatment of respiratory and gastrointestinal diseases ROCHE PALO ALTO LLC (US) 2011-08-30 US disclosed