SCHEMBL12376924

SCHEMBL12376924

N=C(N)CCCc1ccc(CCC(=N)N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.43
NPC1 O15118 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
RAB9A P51151 1/20 0.43
HIF1A Q16665 1/20 0.43
BLM P54132 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HDAC1 Q13547 4/20 0.39
HDAC3 O15379 1/20 0.39
MAPK1 P28482 1/20 0.39
ADRA1A P35348 1/20 0.39
HDAC4 P56524 1/20 0.39
SLC6A3 Q01959 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13819007 0.95 NOS1 (0.46) NOS1NPC1CYP3A4CYP2D6RAB9A
SCHEMBL12401897 0.93 NOS1 (0.45) NOS1NPC1CYP3A4CYP2D6RAB9A
SCHEMBL12401872 0.91 CYP3A4 (0.43) NOS1NPC1CYP3A4CYP2D6RAB9A
SCHEMBL8780954 0.91 NOS1 (0.50) NOS1NPC1CYP3A4CYP2D6RAB9A
SCHEMBL13537270 0.87 ESR1 (0.52) CYP3A4HIF1ABLMSLC6A3HSD17B10
SCHEMBL10308996 0.87 NOS1 (0.41) NOS1NPC1CYP3A4CYP2D6RAB9A
SCHEMBL5645511 0.85 IDO1 (0.50) IDO1
SCHEMBL21485091 0.84 NOS1 (0.58) NOS1NPC1RAB9AHDAC1HDAC3
Hydrochloric Acid SCHEMBL4717388 0.84 IDO1 (0.52) IDO1
Hydrochloric Acid SCHEMBL1625456 0.83 NOS1 (0.56) NOS1NPC1RAB9AHDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003633-B1 Anti-cancer compositions and methods THE PENN STATE RESEARCH FOUNDATION (US) 2011-08-23 US disclosed