SCHEMBL12377970

SCHEMBL12377970

C=C(C)OC(=O)Nc1ncc(C(N[S@@+]([O-])C(C)(C)C)c2ccc(F)cc2Cl)s1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
CDK5 Q00535 1/20 0.33
FFAR2 O15552 2/20 0.31
MDM2 Q00987 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12377347 1.00 CCNE1 (0.33) CCNE1CDK2CDK5FFAR2MDM2
SCHEMBL14145695 0.90 CCNE1 (0.34) CCNE1CDK2CDK5MDM2
SCHEMBL14145694 0.90 CCNE1 (0.34) CCNE1CDK2CDK5MDM2
SCHEMBL1691012 0.89 LCK (0.35) CCNE1CDK2CDK5FFAR2MDM2
SCHEMBL1691316 0.89 LCK (0.35) CCNE1CDK2CDK5FFAR2MDM2
SCHEMBL1926160 0.89 LCK (0.35) CCNE1CDK2CDK5FFAR2MDM2
SCHEMBL10124744 0.89 LCK (0.35) CCNE1CDK2CDK5FFAR2MDM2
SCHEMBL10125058 0.89 LCK (0.35) CCNE1CDK2CDK5FFAR2MDM2
SCHEMBL16681690 0.89 LCK (0.35) CCNE1CDK2CDK5FFAR2MDM2
SCHEMBL12377971 0.88 FFAR2 (0.35) CCNE1CDK2CDK5FFAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999113-B2 Such as 1-(benzo[d][1,3]dioxol-6-yl)-n-(5-((2-chlorophenyl)(3-hydroxypyrrolidin-1-yl)methyl)thiazol-2-yl)cyclopropanecarboxamide; genetic disorders VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-08-16 US disclosed