SCHEMBL12377971

SCHEMBL12377971

C=C(C)OC(=O)Nc1ncc(C(N[S@+]([O-])C(C)(C)C)c2ccc(Cl)cc2F)s1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FFAR2 O15552 9/20 0.35
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
CDK5 Q00535 1/20 0.33
CYP3A4 P08684 4/20 0.32
CYP3A5 P20815 4/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
PYGL P06737 1/20 0.31
S1PR3 Q99500 2/20 0.31
GRM4 Q14833 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1923732 0.89 S1PR3 (0.39) FFAR2CCNE1CDK2CDK5CYP3A4
SCHEMBL1690967 0.89 S1PR3 (0.39) FFAR2CCNE1CDK2CDK5CYP3A4
SCHEMBL10125038 0.89 S1PR3 (0.39) FFAR2CCNE1CDK2CDK5CYP3A4
SCHEMBL1924081 0.89 S1PR3 (0.39) FFAR2CCNE1CDK2CDK5CYP3A4
SCHEMBL1690804 0.89 S1PR3 (0.39) FFAR2CCNE1CDK2CDK5CYP3A4
SCHEMBL12377970 0.88 CCNE1 (0.33) FFAR2CCNE1CDK2CDK5
SCHEMBL12377347 0.88 CCNE1 (0.33) FFAR2CCNE1CDK2CDK5
SCHEMBL16678081 0.87 FFAR2 (0.38) FFAR2CCNE1CDK2CDK5MAPT
SCHEMBL4765079 0.85 SMN1; SMN2 (0.41) FFAR2
SCHEMBL14145310 0.83 S1PR3 (0.37) FFAR2CCNE1CDK2CDK5CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999113-B2 Such as 1-(benzo[d][1,3]dioxol-6-yl)-n-(5-((2-chlorophenyl)(3-hydroxypyrrolidin-1-yl)methyl)thiazol-2-yl)cyclopropanecarboxamide; genetic disorders VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-08-16 US disclosed