SCHEMBL12390334

SCHEMBL12390334

Cc1ccc(Cn2c(-c3ccc(C(=O)N4CCNCC4)cc3)cc(C(F)(F)F)c(N)c2=O)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.41
GRIN2B Q13224 2/20 0.40
ATR Q13535 5/20 0.38
HPGD P15428 1/20 0.36
CCNC P24863 2/20 0.36
CDK8 P49336 2/20 0.36
RAD52 P43351 1/20 0.36
UBE2N P61088 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
GABRA4 P48169 1/20 0.35
ABL1 P00519 2/20 0.35
BCR P11274 2/20 0.35
KDM1A O60341 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12390414 0.91 GRIN2B (0.46) GRIN2BHPGDKDM1A
SCHEMBL12390628 0.88 RXRA (0.44) KCNH2GRIN2BATRHPGDCCNC
SCHEMBL12366784 0.88 GRIN2B (0.41) KCNH2GRIN2BATRHPGDCCNC
Hydrochloric Acid SCHEMBL2268439 0.88 RXRA (0.44) KCNH2GRIN2BATRHPGDCCNC
SCHEMBL12390411 0.86 GRIN2B (0.40) GRIN2BABL1BCRKDM1A
SCHEMBL12390420 0.85 ALDH1A1 (0.40) GRIN2B
SCHEMBL12390195 0.82 MAPT (0.42)
SCHEMBL12390408 0.80 F2 (0.38)
SCHEMBL2262542 0.80 RXRA (0.46) GRIN2BHPGDKDM1A
SCHEMBL12366778 0.79 GRIN2B (0.46) GRIN2BHPGDKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed