SCHEMBL1241635

SCHEMBL1241635

CCCC=Cc1ccc2ccc[c]c2c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.38
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
ALDH1A1 P00352 1/20 0.34
GLA P06280 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
RELA Q04206 1/20 0.33
NQO2 P16083 2/20 0.31
GABBR2 O75899 1/20 0.30
GABBR1 Q9UBS5 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA7 P36544 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL294273 0.88 TLR8 (0.38) TLR8HDAC1HDAC8ALDH1A1GLA
SCHEMBL294272 0.88 TLR8 (0.38) TLR8HDAC1HDAC8ALDH1A1GLA
SCHEMBL5748128 0.73 CYP2A6 (0.39) ALDH1A1
SCHEMBL7790790 0.73 ALDH1A1 (0.37) ALDH1A1RELA
SCHEMBL28422917 0.72 TLR8 (0.32) TLR8
SCHEMBL28424989 0.70 TLR8 (0.33) TLR8
SCHEMBL8625941 0.70 CNR1 (0.39)
Anthracene SCHEMBL28105538 0.69 TLR8 (0.47) TLR8RELA
SCHEMBL5748073 0.69 CYP1A2 (0.53) ALDH1A1MAPTSMN1; SMN2
SCHEMBL29084182 0.69 HDAC1 (0.56) HDAC1HDAC8ALDH1A1GLAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-B9 HETEROCYCLIC COMPOUND OTSUKA PHARMA CO LTD (JP) 2012-01-18 EP disclosed
EP-1919907-B1 HETEROCYCLIC COMPOUND OTSUKA PHARMA CO LTD (JP) 2011-02-23 EP disclosed